SCHEMBL5335078

SCHEMBL5335078

Cc1nc(C(F)(F)F)ccc1CC=O

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.38
LMNA P02545 1/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
KDM4E B2RXH2 1/20 0.36
CXCR4 P61073 1/20 0.36
TRPV1 Q8NER1 2/20 0.36
MBOAT4 Q96T53 3/20 0.35
CNR1 P21554 5/20 0.35
CYP3A4 P08684 2/20 0.35
CYP2C9 P11712 2/20 0.35
CYP2C19 P33261 2/20 0.35
NR1H2 P55055 1/20 0.34
NR1H3 Q13133 1/20 0.34
TKT P29401 1/20 0.33
BCHE P06276 1/20 0.32
ACHE P22303 1/20 0.32
P2RX7 Q99572 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5265318 0.82 LMNA (0.40) GAALMNANPC1RAB9AKDM4E
SCHEMBL19616101 0.79 TRPV1 (0.35) LMNATRPV1P2RX7
SCHEMBL23269412 0.78 LMNA (0.40) GAALMNANPC1RAB9AKDM4E
SCHEMBL2870247 0.77 KDM4E (0.39) GAALMNANPC1RAB9AKDM4E
SCHEMBL4484041 0.77 KDM4E (0.39) GAALMNANPC1RAB9AKDM4E
SCHEMBL2866080 0.77 TKT (0.40) GAALMNANPC1RAB9AKDM4E
SCHEMBL404270 0.77 KDM4E (0.39) GAALMNANPC1RAB9AKDM4E
SCHEMBL21503616 0.75 KDM4E (0.38) GAALMNANPC1RAB9AKDM4E
SCHEMBL19771944 0.75 KDM4E (0.38) GAALMNANPC1RAB9AKDM4E
SCHEMBL3558234 0.75 MBOAT4 (0.49) GAALMNANPC1RAB9AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012068210-A1 PYRIDYL-THIAZOLYL INHIBITORS OF PRO-MATRIX METALLOPROTEINASE ACTIVATION JANSSEN PHARMACEUTICA NV (BE) 2012-05-24 WO disclosed
EP-1824828-A2 PYRIDINE BASED COMPOUNDS USEFUL AS INTERMEDIATES FOR PHARMACEUTICAL OR AGRICULTURAL END-PRODUCTS Peakdale Molecular Limited (GB) 2007-08-29 EP disclosed
WO-2006059103-A2 PYRIDINE BASED COMPOUNDS USEFUL AS INTERMEDIATES FOR PHARMACEUTICAL OR AGRICULTURAL END-PRODUCTS PEAKDALE MOLECULAR LIMITED (GB) 2006-06-08 WO disclosed