SCHEMBL5337520

SCHEMBL5337520

CC1=C(C(=O)OCC(C)C)C(c2cccc(Br)c2)NC(=O)N1

nearest known ligand 0.72

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.66
ADORA2B P29275 4/20 0.64
ADORA1 P30542 1/20 0.64
MCL1 Q07820 1/20 0.64
KIF11 P52732 1/20 0.61
PKM P14618 1/20 0.55
MEN1 O00255 1/20 0.53
KMT2A Q03164 1/20 0.53
POLB P06746 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5352781 0.89 KIF11 (0.77) ADORA2BKIF11PKM
SCHEMBL5345378 0.87 MAPT (0.66) MAPTADORA2BADORA1MCL1KIF11
SCHEMBL5352815 0.86 KIF11 (0.65) ADORA2BKIF11PKMMEN1KMT2A
SCHEMBL10113135 0.85 GAA (0.64) ADORA2BKIF11PKMMEN1KMT2A
SCHEMBL10113145 0.83 HSD17B10 (0.67) ADORA2BKIF11PKMMEN1KMT2A
SCHEMBL10144746 0.83 POLB (0.61) KIF11PKMPOLB
SCHEMBL5343438 0.82 POLB (0.63) KIF11PKMPOLB
SCHEMBL10113224 0.82 MAPT (0.82) MAPTADORA2BADORA1MCL1POLB
SCHEMBL10113437 0.81 ADORA2B (0.61) ADORA2BKIF11PKMMEN1KMT2A
SCHEMBL16457636 0.81 TSHR (0.70) PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007101213-A2 NOVEL 2-OXO-1,2,3,4-TETRAHYDROPYRIMIDINES, BICYCLIC PYRIMIDINE DIONES AND IMIDAZOLIDINE-2,4-DIONES USEFUL AS INDUCIBLE NITRIC OXIDE SYNTHASE INHIBITORS KALYPSYS, INC. (US) 2007-09-07 WO disclosed