SCHEMBL5338757

SCHEMBL5338757

Cc1ccc(C(=O)N(C)C(N)=O)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.48
CES2 O00748 3/20 0.48
CES1 P23141 3/20 0.48
LMNA P02545 2/20 0.48
SMN1; SMN2 Q16637 3/20 0.46
PKM P14618 2/20 0.43
HTT P42858 2/20 0.43
ATM Q13315 2/20 0.43
NPSR1 Q6W5P4 2/20 0.43
TDP1 Q9NUW8 2/20 0.43
HPGD P15428 2/20 0.43
NLRP1 Q9C000 1/20 0.43
GAA P10253 1/20 0.43
MEN1 O00255 1/20 0.43
NTSR1 P30989 1/20 0.43
KMT2A Q03164 1/20 0.43
ALOX5 P09917 1/20 0.43
SRD5A2 P31213 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11692698 0.84 ALDH1A1 (0.45) ALDH1A1CES2CES1LMNASMN1; SMN2
SCHEMBL7104370 0.81 MAPT (0.50) ALDH1A1CES2CES1TDP1HPGD
SCHEMBL27383304 0.81 ALDH1A1 (0.54) ALDH1A1CES2CES1LMNASMN1; SMN2
SCHEMBL11464381 0.81 MAPT (0.50) ALDH1A1CES2CES1TDP1HPGD
Hydrochloric Acid SCHEMBL4562959 0.79 MAPT (0.48) ALDH1A1CES2CES1TDP1HPGD
SCHEMBL11685910 0.79 ALDH1A1 (0.48) ALDH1A1CES2CES1LMNASMN1; SMN2
Hydrochloric Acid SCHEMBL11685915 0.79 ALDH1A1 (0.52) ALDH1A1CES2CES1LMNASMN1; SMN2
SCHEMBL11216329 0.78 ALDH1A1 (0.56) ALDH1A1CES2CES1LMNASMN1; SMN2
SCHEMBL469413 0.78 ALDH1A1 (0.61) ALDH1A1CES2CES1LMNASMN1; SMN2
SCHEMBL3246852 0.78 KDM4E (0.53) ALDH1A1LMNASMN1; SMN2HTTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1753731-A2 PYRIMIDIN-4-ONE DERIVATIVES AND THEIR USE AS P38 KINASE MODULATORS Pharmacia Corporation (US) 2007-02-21 EP disclosed
WO-2004087677-A2 PYRIMIDIN-4-ONE DERIVATIVES AND THEIR USE AS P38 KINASE MODULATORS PHARMACIA CORPORATION (US) 2004-10-14 WO disclosed