SCHEMBL5340893

SCHEMBL5340893

Cc1cc(C2CCCN2C(CC2=COCO2)(Cc2ccccc2)C(N)=O)nc(-n2ccnc2)n1

nearest known ligand 0.48

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 18/20 0.48
NOS1 P29475 4/20 0.48
KDM4E B2RXH2 1/20 0.33
TSHR P16473 1/20 0.33
MAPK1 P28482 1/20 0.33
ATM Q13315 1/20 0.33
TDP1 Q9NUW8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3560184 0.77 NOS2 (0.53) NOS2NOS1
SCHEMBL3569388 0.75 NOS2 (0.60) NOS2NOS1TSHR
Hydrochloric Acid SCHEMBL3571851 0.74 NOS2 (0.60) NOS2NOS1TSHR
SCHEMBL3562923 0.73 NOS2 (0.58) NOS2NOS1TSHR
SCHEMBL5340887 0.73 NOS2 (0.61) NOS2NOS1
SCHEMBL3556108 0.71 NOS1 (0.55) NOS2NOS1KDM4ETSHRMAPK1
SCHEMBL3566595 0.70 NOS2 (0.59) NOS2NOS1KDM4ETSHRMAPK1
SCHEMBL3561935 0.69 NOS2 (0.51) NOS2NOS1
SCHEMBL5340900 0.67 NOS2 (0.65) NOS2NOS1
SCHEMBL4884982 0.67 NOS2 (0.61) NOS2NOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007062417-A1 METHODS OF PREPARING 2-IMIDAZOL-1-YL-4-METHYL-6-PYRROLIDIN-2-YL-PYRIMIDINE AND 4-(1-ALKYLPYRROLIDIN-2-YL)-2-(1H-IMIDAZOL-1-YL)-6-METHYLPYRIMIDINE DERIVATIVES KALYPSYS, INC. (US) 2007-05-31 WO disclosed