SCHEMBL5340948

SCHEMBL5340948

O=C(c1cc(Cl)c2nc(-c3ccccc3Cl)c(-c3ccc(Cl)cc3)n2c1)N1CCOCC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPAS1 Q99814 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C19 P33261 1/20 0.46
PHGDH O43175 1/20 0.46
GAA P10253 1/20 0.46
HTR2C P28335 1/20 0.45
PKM P14618 2/20 0.44
ALDH1A1 P00352 2/20 0.44
AKT1 P31749 2/20 0.44
AKT2 P31751 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.43
KDM4E B2RXH2 2/20 0.43
HPGD P15428 2/20 0.43
NPC1 O15118 1/20 0.43
TP53 P04637 1/20 0.43
MAPK1 P28482 1/20 0.43
RAB9A P51151 1/20 0.43
CYP1A2 P05177 1/20 0.43
CNR1 P21554 1/20 0.42
AKR1C3 P42330 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5337506 0.90 PHGDH (0.51) CYP3A4CYP2C19PHGDHGAAPKM
SCHEMBL5336841 0.82 SMN1; SMN2 (0.47) CYP3A4CYP2C19PHGDHGAAPKM
SCHEMBL5351210 0.81 CNR1 (0.54) AKT1AKT2HPGDNPC1RAB9A
SCHEMBL5342230 0.80 CNR1 (0.56) AKT1AKT2HPGDNPC1RAB9A
SCHEMBL5335702 0.78 POLB (0.51) CYP3A4ALDH1A1AKT1AKT2TP53
SCHEMBL5343352 0.77 AKT1 (0.49) CYP3A4CYP2C19ALDH1A1AKT1AKT2
SCHEMBL5341020 0.76 AKT1 (0.50) AKT1AKT2CNR1
SCHEMBL5380026 0.75 GABRA2 (0.49) CYP3A4AKT1AKT2TP53CNR1
SCHEMBL5342400 0.74 AKT1 (0.50) CYP3A4AKT1AKT2APC
SCHEMBL5317129 0.74 AKT1 (0.48) AKT1AKT2SMN1; SMN2KDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007086080-A2 NOVEL IMIDAZO[1,2-a]PYRIDINE CANNABINOID RECEPTOR LIGANDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM GLENMARK PHARMACEUTICALS LIMITED (IN) 2007-08-02 WO claimed
WO-2007086080-A2 NOVEL IMIDAZO[1,2-a]PYRIDINE CANNABINOID RECEPTOR LIGANDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM GLENMARK PHARMACEUTICALS LIMITED (IN) 2007-08-02 WO disclosed