SCHEMBL5341989

SCHEMBL5341989

CCOC(=O)n1c(CNC(=O)OC(C)(C)C)ccc1-c1ccnc(N)n1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 2/20 0.39
DBF4 Q9UBU7 1/20 0.39
MAPKAPK2 P49137 5/20 0.36
JAK2 O60674 3/20 0.36
L3MBTL1 Q9Y468 1/20 0.35
MAPK14 Q16539 1/20 0.35
HSP90AA1 P07900 1/20 0.35
HSP90AB1 P08238 1/20 0.35
BTK Q06187 1/20 0.35
AAK1 Q2M2I8 1/20 0.34
KDM4A O75164 1/20 0.33
BRD4 O60885 1/20 0.33
CSNK2A2 P19784 1/20 0.33
CSNK2A1 P68400 1/20 0.33
ADORA3 P0DMS8 1/20 0.33
ADORA2A P29274 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5341992 0.72 JAK2 (0.47) CDC7DBF4JAK2CSNK2A1
SCHEMBL16793748 0.71 BTK (0.63) BTKAAK1
SCHEMBL15074549 0.69 CDC7 (0.55) CDC7DBF4JAK2ADORA3ADORA2A
SCHEMBL14007210 0.67 AKT3 (0.55) L3MBTL1BTK
SCHEMBL3336071 0.66 HRH4 (0.60)
SCHEMBL29631866 0.65 KDM4A (0.43) MAPKAPK2L3MBTL1KDM4A
SCHEMBL19013326 0.65 KDM4A (0.43) MAPKAPK2L3MBTL1KDM4A
SCHEMBL3778944 0.64 HRH3 (0.59) BRD4ADORA2A
SCHEMBL509487 0.63 KDM5B (0.53) BRD4
SCHEMBL31627088 0.63 NPSR1 (0.45) BRD4ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007096334-A1 PYRROLOPYRROLONES ACTIVE AS KINASE INHIBITORS PFIZER ITALIA SRL (IT) 2007-08-30 WO claimed