SCHEMBL534417

SCHEMBL534417

CC(C)(C)OC(=O)NC(C(=O)O)c1cccc(C(Cc2ccc(Br)cc2)NS(=O)(=O)c2cccnc2)n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSS P25774 1/20 0.40
CTSK P43235 1/20 0.40
CYP3A4 P08684 8/20 0.39
PTPRB P23467 5/20 0.39
SLC1A3 P43003 1/20 0.38
SLC1A2 P43004 1/20 0.38
SLC1A1 P43005 1/20 0.38
ALDH1A1 P00352 2/20 0.37
LMNA P02545 2/20 0.37
PKM P14618 2/20 0.37
HPGD P15428 2/20 0.37
TSHR P16473 2/20 0.37
HTT P42858 2/20 0.37
NPSR1 Q6W5P4 2/20 0.37
HSD17B10 Q99714 2/20 0.37
TP53 P04637 1/20 0.37
MAPT P10636 1/20 0.37
AGTR1 P30556 1/20 0.37
RAB9A P51151 1/20 0.37
MEN1 O00255 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL534415 0.82 CTSS (0.36) CTSSCTSKCYP3A4PTPRBKMT2A
SCHEMBL533795 0.81 SLC1A3 (0.35) CTSSPTPRBSLC1A3SLC1A2SLC1A1
SCHEMBL3459165 0.81 PTGER2 (0.38) SLC1A3SLC1A2SLC1A1KMT2AADAM17
SCHEMBL534416 0.80 PTGER2 (0.57) PTGER2
SCHEMBL6519267 0.79 PTGER2 (0.34) CTSSSLC1A3SLC1A2SLC1A1KMT2A
SCHEMBL6519253 0.77 SLC1A3 (0.34) CTSSSLC1A3SLC1A2SLC1A1KMT2A
SCHEMBL534320 0.73 PTGER2 (0.38) PTPRBSLC1A3SLC1A2SLC1A1BCL2
SCHEMBL12982541 0.73 PTGER2 (0.53) PTGER2
SCHEMBL533647 0.73 PTGER2 (0.41) PTPRBBCL2PTGER2
SCHEMBL10322183 0.73 PTPRB (0.35) PTPRBSLC1A3SLC1A2SLC1A1ADAM17

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2415763-A1 PHARMACEUTICAL COMPOSITION FOR TREATING OR PREVENTING GLAUCOMA Ube Industries, Ltd. (JP) 2012-02-08 EP disclosed