SCHEMBL5344446

SCHEMBL5344446

CCOC(=O)C1=C(C)NC(=O)NC1c1cccc(-c2cccnc2)c1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 1/20 0.67
ALDH1A1 P00352 2/20 0.56
GAA P10253 2/20 0.54
ADORA2B P29275 3/20 0.53
MAPK1 P28482 3/20 0.53
HSD17B10 Q99714 2/20 0.53
CYP1A2 P05177 1/20 0.53
CYP2C9 P11712 1/20 0.53
CYP2C19 P33261 1/20 0.53
TSHR P16473 1/20 0.53
RAB9A P51151 1/20 0.53
PKM P14618 1/20 0.52
KDM4E B2RXH2 1/20 0.52
HPGD P15428 1/20 0.52
CASP1 P29466 1/20 0.52
CASP7 P55210 1/20 0.52
CA12 O43570 1/20 0.52
CA1 P00915 1/20 0.52
CA2 P00918 1/20 0.52
CA7 P43166 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5351543 0.88 KIF11 (0.66) KIF11ALDH1A1GAAADORA2BMAPK1
SCHEMBL7267796 0.84 CACNA1F (0.57) ALDH1A1GAAMAPK1HSD17B10CYP1A2
SCHEMBL31705192 0.81 KIF11 (0.80) KIF11ALDH1A1GAAADORA2BMAPK1
SCHEMBL5340534 0.81 KIF11 (0.80) KIF11ALDH1A1GAAADORA2BMAPK1
SCHEMBL5341216 0.80 KIF11 (1.00) KIF11ALDH1A1GAAADORA2BMAPK1
SCHEMBL5351765 0.79 KIF11 (0.77) KIF11ALDH1A1GAAADORA2BMAPK1
SCHEMBL5354452 0.79 PKM (0.78) KIF11ALDH1A1GAAADORA2BMAPK1
SCHEMBL5352781 0.79 KIF11 (0.77) KIF11ALDH1A1GAAADORA2BMAPK1
SCHEMBL14413847 0.79 KIF11 (0.77) KIF11ALDH1A1GAAADORA2BMAPK1
SCHEMBL19752682 0.79 PKM (0.78) KIF11ALDH1A1GAAADORA2BMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007101213-A2 NOVEL 2-OXO-1,2,3,4-TETRAHYDROPYRIMIDINES, BICYCLIC PYRIMIDINE DIONES AND IMIDAZOLIDINE-2,4-DIONES USEFUL AS INDUCIBLE NITRIC OXIDE SYNTHASE INHIBITORS KALYPSYS, INC. (US) 2007-09-07 WO disclosed
WO-2007101213-A2 NOVEL 2-OXO-1,2,3,4-TETRAHYDROPYRIMIDINES, BICYCLIC PYRIMIDINE DIONES AND IMIDAZOLIDINE-2,4-DIONES USEFUL AS INDUCIBLE NITRIC OXIDE SYNTHASE INHIBITORS KALYPSYS, INC. (US) 2007-09-07 WO disclosed