SCHEMBL5346776

SCHEMBL5346776

Oc1ccc(-c2c(-c3ccc(Cl)cc3)nc3ncc(-c4cccc(C(F)(F)F)c4)cn23)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 1/20 0.42
AKT2 P31751 1/20 0.42
MAPT P10636 2/20 0.39
GAA P10253 1/20 0.39
ADORA2A P29274 1/20 0.39
ADORA1 P30542 1/20 0.39
USP7 Q93009 2/20 0.38
CCNA2 P20248 1/20 0.38
CDK2 P24941 1/20 0.38
CDK5 Q00535 1/20 0.38
DYRK1A Q13627 1/20 0.38
CDK5R1 Q15078 1/20 0.38
DYRK2 Q92630 1/20 0.38
DYRK1B Q9Y463 1/20 0.38
GRIN2B Q13224 5/20 0.37
MAOB P27338 1/20 0.37
FYN P06241 1/20 0.37
GRIN1 Q05586 1/20 0.37
KDM4E B2RXH2 1/20 0.37
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5338540 0.95 AKT1 (0.46) AKT1AKT2GAAADORA2AADORA1
Hydrochloric Acid SCHEMBL5344599 0.94 AKT1 (0.45) AKT1AKT2GAAADORA2AADORA1
SCHEMBL5319387 0.87 AKT1 (0.41) AKT1AKT2MAPTGAAADORA2A
SCHEMBL5343644 0.87 GRIN1 (0.46) AKT1AKT2MAPTGAAGRIN2B
SCHEMBL5343214 0.85 TDP1 (0.47) AKT1AKT2MAPTGAAADORA2A
SCHEMBL5322231 0.85 AKT1 (0.48) AKT1AKT2GAAADORA1FYN
SCHEMBL5340690 0.83 MAOB (0.40) MAPTGAAADORA2AADORA1CCNA2
SCHEMBL5324596 0.83 TDP1 (0.46) AKT1AKT2GAAADORA2AADORA1
SCHEMBL5341386 0.82 AKT1 (0.49) AKT1AKT2GAAKDM4ELMNA
SCHEMBL5325683 0.81 AKT1 (0.51) AKT1AKT2MAPTGAAADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007096764-A2 BICYCLIC HETEROARYL DERIVATIVES AS CANNABINOID RECEPTOR MODULATORS GLENMARK PHARMACEUTICALS S.A. (US) 2007-08-30 WO claimed
WO-2007096764-A2 BICYCLIC HETEROARYL DERIVATIVES AS CANNABINOID RECEPTOR MODULATORS GLENMARK PHARMACEUTICALS S.A. (US) 2007-08-30 WO disclosed