SCHEMBL534838

SCHEMBL534838

COc1cc(C#N)ccc1CN(C)CC(=O)O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.45
KDM4E B2RXH2 4/20 0.45
POLB P06746 2/20 0.44
SMN1; SMN2 Q16637 4/20 0.44
HTT P42858 3/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
NPSR1 Q6W5P4 1/20 0.44
LMNA P02545 3/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
TDP1 Q9NUW8 1/20 0.43
PYCR1 P32322 1/20 0.41
CD274 Q9NZQ7 2/20 0.40
PDCD1 Q15116 1/20 0.40
MAPT P10636 1/20 0.40
PLA2G4A P47712 1/20 0.39
LTB4R Q15722 1/20 0.39
PPARD Q03181 1/20 0.39
PPARA Q07869 1/20 0.39
AR P10275 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27001733 0.89 ALDH1A1 (0.41) ALDH1A1KDM4EPOLBMEN1KMT2A
SCHEMBL410797 0.84 ABCB1 (0.41) ALDH1A1KDM4EPOLBSMN1; SMN2HTT
SCHEMBL534824 0.81 NPSR1 (0.60) ALDH1A1POLBHTTNPSR1PYCR1
SCHEMBL2773430 0.80 HTT (0.46) ALDH1A1KDM4EPOLBHTTMEN1
SCHEMBL27001732 0.76 ABCB1 (0.42) ALDH1A1KDM4EPOLBMAPTPLA2G4A
SCHEMBL1855982 0.75 AR (0.49) HTTMAPTPLA2G4ALTB4RAR
SCHEMBL13098166 0.75 AR (0.43) POLBPYCR1ARMAOB
SCHEMBL26144386 0.74 CETP (0.38) LMNAMAPTPLA2G4ALTB4RAR
SCHEMBL23201206 0.74 ABCB1 (0.39) ALDH1A1KDM4EPOLBMAPTPLA2G4A
SCHEMBL14183081 0.74 POLB (0.59) POLBHTTMEN1KMT2ANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2414341-A2 OXADIAZOLE DERIVATIVES Merck Serono SA (CH) 2012-02-08 EP disclosed
WO-2010115751-A2 OXADIAZOLE DERIVATIVES MERCK SERONO S.A. (CH) 2010-10-14 WO disclosed