SCHEMBL534824

SCHEMBL534824

CN(CC(=O)O)Cc1ccc(C#N)cc1Cl

nearest known ligand 0.60

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.60
HTT P42858 1/20 0.60
HIF1A Q16665 1/20 0.45
ALDH1A1 P00352 2/20 0.44
POLB P06746 1/20 0.43
P2RX7 Q99572 3/20 0.42
PYCR1 P32322 2/20 0.40
PDK1 Q15118 1/20 0.40
PDK2 Q15119 1/20 0.40
PDK3 Q15120 1/20 0.40
PDK4 Q16654 1/20 0.40
CYP19A1 P11511 1/20 0.39
EPHX2 P34913 1/20 0.39
FFAR1 O14842 1/20 0.38
MRGPRX4 Q96LA9 2/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.38
PDCD1 Q15116 1/20 0.37
CD274 Q9NZQ7 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5110282 0.83 HTT (0.50) NPSR1HTTALDH1A1POLBP2RX7
SCHEMBL403900 0.82 HTT (0.54) NPSR1HTTALDH1A1POLBP2RX7
SCHEMBL2773430 0.82 HTT (0.46) NPSR1HTTHIF1AALDH1A1POLB
SCHEMBL534838 0.81 ALDH1A1 (0.45) NPSR1HTTALDH1A1POLBPYCR1
SCHEMBL30349567 0.77 ALDH1A1 (0.50) NPSR1HTTALDH1A1P2RX7PDK1
SCHEMBL14660970 0.77 ALDH1A1 (0.50) NPSR1HTTALDH1A1P2RX7PDK1
SCHEMBL14183081 0.76 POLB (0.59) NPSR1HTTPOLB
SCHEMBL11112081 0.75 FFAR1 (0.51) ALDH1A1P2RX7FFAR1MRGPRX4
SCHEMBL2773568 0.74 MEP1A (0.57) PDK1FFAR1PDCD1CD274
SCHEMBL5912934 0.74 HTT (0.45) NPSR1HTTALDH1A1P2RX7PDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2414341-A2 OXADIAZOLE DERIVATIVES Merck Serono SA (CH) 2012-02-08 EP disclosed
WO-2010115751-A2 OXADIAZOLE DERIVATIVES MERCK SERONO S.A. (CH) 2010-10-14 WO disclosed