SCHEMBL5350376

SCHEMBL5350376

O=S(=O)(c1ccccc1Cl)N1CCCN(c2c(Cl)cccc2Cl)CC1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 7/20 0.63
TSHR P16473 2/20 0.55
KMT2A Q03164 3/20 0.53
LMNA P02545 1/20 0.53
MAPT P10636 2/20 0.52
MAPK1 P28482 2/20 0.52
CYP3A4 P08684 2/20 0.51
CYP2C9 P11712 2/20 0.51
CYP2C19 P33261 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.49
CHRM2 P08172 1/20 0.48
CHRM5 P08912 1/20 0.48
CHRM1 P11229 1/20 0.48
CHRM3 P20309 1/20 0.48
GBA1 P04062 1/20 0.48
MEN1 O00255 2/20 0.47
TP53 P04637 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2D6 P10635 1/20 0.46
NFKB1 P19838 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3223553 0.94 CHRM4 (0.61) CHRM4TSHRMAPTMAPK1CYP3A4
SCHEMBL5347507 0.89 CHRM4 (0.61) CHRM4TSHRKMT2ALMNAMAPT
SCHEMBL5331434 0.87 CHRM4 (0.64) CHRM4TSHRKMT2ALMNAMAPT
SCHEMBL3210281 0.82 CHRM4 (0.59) CHRM4TSHRCYP3A4CHRM2CHRM5
SCHEMBL10723724 0.82 CHRM4 (0.64) CHRM4TSHRKMT2ALMNAMAPT
SCHEMBL31684034 0.81 TSHR (0.78) CHRM4TSHRKMT2ALMNAMAPT
SCHEMBL4555453 0.81 TSHR (0.78) CHRM4TSHRKMT2ALMNAMAPT
SCHEMBL2961026 0.80 CHRM4 (0.62) CHRM4TSHRKMT2ALMNAMAPT
SCHEMBL5329287 0.79 MEN1 (0.60) CHRM4TSHRKMT2ALMNAMAPT
SCHEMBL2962429 0.78 MEN1 (0.62) CHRM4KMT2ALMNASMN1; SMN2GBA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007122411-A1 DIAZEPAN-1-YL-SULFONYL DERIVATIVES FOR THE TREATMENT OF METABOLIC SYNDROME ASTRAZENECA AB (SE) 2007-11-01 WO claimed