SCHEMBL5350906

SCHEMBL5350906

Cc1cc2c(cc1C=Cc1ccccc1)C(C1CCCCC1)=NN(C)C(=O)N2c1ccc(CC2=NCCN2)cc1

nearest known ligand 0.55

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTH1R Q03431 19/20 0.55
LMNA P02545 1/20 0.34
CYP1A2 P05177 1/20 0.34
ADRA2A P08913 1/20 0.34
CYP2D6 P10635 1/20 0.34
TSHR P16473 1/20 0.34
ADRA2B P18089 1/20 0.34
ADRA2C P18825 1/20 0.34
ADRA1D P25100 1/20 0.34
ADRA1A P35348 1/20 0.34
ADRA1B P35368 1/20 0.34
TAAR1 Q96RJ0 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5350903 1.00 PTH1R (0.55) PTH1RLMNACYP1A2ADRA2ACYP2D6
SCHEMBL5352412 0.85 PTH1R (0.56) PTH1RLMNACYP1A2ADRA2ACYP2D6
SCHEMBL5349639 0.85 PTH1R (0.47) PTH1R
SCHEMBL5349636 0.85 PTH1R (0.47) PTH1R
SCHEMBL5353466 0.84 PTH1R (0.54) PTH1R
SCHEMBL5359824 0.82 PTH1R (0.67) PTH1R
SCHEMBL5368169 0.76 PTH1R (0.69) PTH1RLMNACYP1A2ADRA2ACYP2D6
SCHEMBL5356554 0.75 PTH1R (0.67) PTH1R
SCHEMBL5324368 0.75 PTH1R (0.67) PTH1RLMNACYP1A2ADRA2ACYP2D6
SCHEMBL5350640 0.74 PTH1R (0.66) PTH1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007135417-A1 BENZOTRIAZEPINONE DERIVATIVES JAMES BLACK FOUNDATION (GB) 2007-11-29 WO disclosed