SCHEMBL5352716

SCHEMBL5352716

O=S(=O)(Cc1ccccc1)NC1CCC(C(O)(C(F)(F)F)C(F)(F)F)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.43
ADRA1D P25100 1/20 0.43
ADRA1A P35348 1/20 0.43
ADRA1B P35368 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
MMP1 P03956 1/20 0.43
MMP2 P08253 1/20 0.43
MMP9 P14780 1/20 0.43
MMP8 P22894 1/20 0.43
MMP13 P45452 1/20 0.43
LIPE Q05469 2/20 0.40
F2R P25116 1/20 0.39
RORC P51449 1/20 0.38
KMT2A Q03164 1/20 0.38
NR1H2 P55055 1/20 0.37
STS P08842 1/20 0.37
FAAH O00519 1/20 0.36
PRSS1 P07477 1/20 0.36
PRSS2 P07478 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4171714 0.83 CA1 (0.55) DRD2ADRA1DADRA1AADRA1BCA1
SCHEMBL5352810 0.80 KDM4E (0.46) KMT2A
SCHEMBL5352814 0.80 KDM4E (0.46) KMT2A
SCHEMBL5366556 0.80 KDM4E (0.46) KMT2A
SCHEMBL5352146 0.77 DRD2 (0.43) DRD2ADRA1DADRA1AADRA1BCA1
SCHEMBL10153507 0.76 F2 (0.48) DRD2ADRA1DADRA1AADRA1BCA1
SCHEMBL4603405 0.76 DRD2 (0.49) DRD2ADRA1DADRA1AADRA1BCA1
SCHEMBL989727 0.75 HSP90AA1 (0.50) DRD2ADRA1DADRA1AADRA1BCA1
SCHEMBL2884267 0.73 CA1 (0.47) DRD2ADRA1DADRA1AADRA1BCA1
SCHEMBL1460750 0.73 RORC (0.50) RORCNR1H2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7253282-B2 Hexafluoroisopropanol substituted cyclohexane derivatives HOFFMAN-LA ROCHE INC. (US) 2007-08-07 US claimed
US-20060135601-A1 Novel hexafluoroisopropanol substituted cyclohexane derivatives HOFFMANN-LA ROCHE INC. 2006-06-22 US claimed
US-7253282-B2 Hexafluoroisopropanol substituted cyclohexane derivatives HOFFMAN-LA ROCHE INC. (US) 2007-08-07 US disclosed
US-20060135601-A1 Novel hexafluoroisopropanol substituted cyclohexane derivatives HOFFMANN-LA ROCHE INC. 2006-06-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060135601-A1 Novel hexafluoroisopropanol substituted cyclohexane derivatives NR1H3, NR1H2, NR1I2 DRD2 1173/4885ADRA1D 56/4885ADRA1A 40/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.