SCHEMBL5354600

SCHEMBL5354600

Cc1ccc(C(N)=O)c(O)c1C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 1/20 0.43
TDP1 Q9NUW8 2/20 0.42
SIRT3 Q9NTG7 1/20 0.42
GRM1 Q13255 1/20 0.41
KDM4E B2RXH2 3/20 0.40
ALDH1A1 P00352 3/20 0.40
MAPT P10636 2/20 0.40
HPGD P15428 2/20 0.40
HSD17B10 Q99714 2/20 0.40
TSHR P16473 1/20 0.40
NNMT P40261 2/20 0.39
KMT2A Q03164 3/20 0.38
MEN1 O00255 1/20 0.38
NPSR1 Q6W5P4 2/20 0.37
MKNK1 Q9BUB5 1/20 0.37
MKNK2 Q9HBH9 1/20 0.37
PKMYT1 Q99640 2/20 0.36
POLB P06746 1/20 0.36
RECQL P46063 1/20 0.36
CLCN2 P51788 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL926767 0.86 ERN1 (0.46) ERN1TDP1SIRT3GRM1KDM4E
SCHEMBL5515911 0.84 ERN1 (0.44) ERN1TDP1SIRT3GRM1KDM4E
SCHEMBL14880244 0.83 MEN1 (0.49) ERN1GRM1KDM4EALDH1A1MAPT
SCHEMBL4132985 0.82 KMT2A (0.46) TDP1GRM1KDM4EALDH1A1MAPT
SCHEMBL354227 0.82 SIRT3 (0.45) TDP1SIRT3KDM4EALDH1A1MAPT
SCHEMBL6667388 0.80 MAPT (0.47) TDP1GRM1KDM4EALDH1A1MAPT
SCHEMBL30149140 0.80 ALDH1A1 (0.57) TDP1GRM1KDM4EALDH1A1MAPT
SCHEMBL317576 0.80 ALDH1A1 (0.57) TDP1GRM1KDM4EALDH1A1MAPT
SCHEMBL32678438 0.80 MAPT (0.47) TDP1GRM1KDM4EALDH1A1MAPT
Hydrochloric Acid SCHEMBL1776795 0.80 SIRT3 (0.44) TDP1SIRT3KDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103626766-B With the synthesis of the heterocyclic fused γ carbolines of substitution 细胞内治疗公司 2017-06-09 CN claimed
WO-2007134421-A1 2-VINYL INDOLES, PYRIDO AND AZEPINO INDOLE DERIVATIVES, 2-ALKYNYL INDOLES, 2-ALKYNYL BENZO[b]FURANS, THEIR PRECURSORS AND NOVEL PROCESSES FOR THE PREPARATION THEREOF LAUTENS MARK (CA) 2007-11-29 WO claimed
CN-113227045-A Synthesis of substituted heterocycle fused gamma-carbolines 细胞内治疗公司 2021-08-06 CN disclosed
CN-113195450-A Synthesis of substituted heterocycle fused gamma-carbolines 细胞内治疗公司 2021-07-30 CN disclosed
CN-110831941-A Synthesis of substituted heterocycle fused gamma-carboline compound 细胞内治疗公司 2020-02-21 CN disclosed
CN-103626766-B With the synthesis of the heterocyclic fused γ carbolines of substitution 细胞内治疗公司 2017-06-09 CN disclosed
CN-101796051-A Synthesis of substituted heterocycle fused gamma-carbolines INTRA CELLULAR THERAPIES INC 2010-08-04 CN disclosed
EP-0154969-A2 Piperazine derivatives and their acid addition salts MITSUBISHI KASEI CORPORATION (JP) 1985-09-18 EP disclosed