SCHEMBL5354891

SCHEMBL5354891

CCCCCc1ccc2c(N)c(C(N)=O)sc2n1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.60
IKBKB O14920 7/20 0.59
LIMK1 P53667 4/20 0.59
RAB9A P51151 8/20 0.51
NPC1 O15118 7/20 0.51
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
POLB P06746 1/20 0.48
KDM4E B2RXH2 5/20 0.48
HSD17B10 Q99714 1/20 0.48
SMN1; SMN2 Q16637 5/20 0.47
HPGD P15428 4/20 0.47
MAPT P10636 4/20 0.47
ALDH1A1 P00352 3/20 0.47
MCL1 Q07820 2/20 0.47
LMNA P02545 1/20 0.47
RECQL P46063 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
CHUK O15111 1/20 0.47
NFKB1 P19838 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL429337 0.91 ADORA2A (0.71) ADORA2AIKBKBLIMK1RAB9ANPC1
SCHEMBL12562456 0.87 ADORA2A (0.62) ADORA2AIKBKBLIMK1RAB9ANPC1
SCHEMBL5326009 0.81 ADORA2A (0.48) ADORA2AIKBKBLIMK1RAB9ANPC1
SCHEMBL26780528 0.81 ADORA2A (0.73) ADORA2AIKBKBLIMK1RAB9ANPC1
SCHEMBL14955421 0.80 ADORA2A (0.75) ADORA2AIKBKBLIMK1RAB9ANPC1
SCHEMBL4657582 0.78 IKBKB (0.93) IKBKBLIMK1RAB9ANPC1POLB
SCHEMBL26784104 0.76 ADORA2A (0.65) ADORA2AIKBKBLIMK1RAB9ANPC1
SCHEMBL16071461 0.75 IKBKB (1.00) IKBKBLIMK1RAB9ANPC1MEN1
SCHEMBL19212248 0.74 ADORA2A (0.60) ADORA2AIKBKBLIMK1RAB9ANPC1
SCHEMBL22957547 0.70 KDM4E (0.67) ADORA2AIKBKBLIMK1RAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006074919-A3 3-AMINO-6-ARYL(OR 6-HETEROARYL)-THIENO[2,3-B]PYRIDIN-2-CARBOXAMIDES, PHARMACEUTICAL PREPARATIONS CONTAINING THE SAME AND THEIR USE AS TNFα INHIBITORS CURACYTE DISCOVERY GMBH (DE) 2007-02-01 WO disclosed
WO-2006074919-A2 3-AMINO-6-ARYL(OR 6-HETEROARYL)-THIENO[2,3-B]PYRIDIN-2-CARBOXAMIDES, PHARMACEUTICAL PREPARATIONS CONTAINING THE SAME AND THEIR USE AS TNFα INHIBITORS CURACYTE DISCOVERY GMBH (DE) 2006-07-20 WO disclosed