SCHEMBL5355164

SCHEMBL5355164

CN(C)CCNS(=O)(=O)c1cc2cc(-c3cc4cc(F)ccc4[nH]c3=O)[nH]c2cc1F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VCP P55072 1/20 0.41
KDR P35968 5/20 0.38
CHEK1 O14757 2/20 0.36
KDM4E B2RXH2 3/20 0.36
PKM P14618 2/20 0.36
TSHR P16473 1/20 0.36
DAO P14920 1/20 0.36
RORC P51449 1/20 0.35
LMNA P02545 2/20 0.35
KLK7 P49862 1/20 0.35
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
RECQL P46063 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HSD17B10 Q99714 1/20 0.34
GAA P10253 1/20 0.34
CDK5 Q00535 1/20 0.34
CDK5R1 Q15078 1/20 0.34
FFAR1 O14842 1/20 0.33
PPARG P37231 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5354824 0.77 KDR (0.56) KDRCHEK1PKMTSHRLMNA
SCHEMBL5359367 0.76 TSHR (0.49) KDRCHEK1KDM4EPKMTSHR
SCHEMBL14625890 0.75 VCP (0.34) VCPKDRKDM4EPKMTSHR
SCHEMBL5368202 0.75 KDR (0.53) VCPKDRCHEK1KDM4EPKM
SCHEMBL5357812 0.74 KDR (0.49) VCPKDRCHEK1KDM4EKLK7
SCHEMBL5367618 0.67 CDK1 (0.47) KDRKDM4ETSHRLMNAALDH1A1
SCHEMBL14590420 0.65 CDK1 (0.45) KDRKDM4EPKMTSHRLMNA
SCHEMBL139863 0.65 KDR (0.59) KDRCHEK1KDM4ELMNAALDH1A1
SCHEMBL1348432 0.65 CYP2C9 (0.50) PKMTSHRKLK7CYP2C9CYP2C19
SCHEMBL5356295 0.64 KDR (0.73) VCPKDRCHEK1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7169788-B2 Tyrosine kinase inhibitors MERCK & CO., INC. (US) 2007-01-30 US disclosed
US-7169788-B2 Tyrosine kinase inhibitors MERCK & CO., INC. (US) 2007-01-30 US disclosed