SCHEMBL5358667

SCHEMBL5358667

O=S1(=O)N=CN(CCF)c2cc(F)ccc21

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.50
TP53 P04637 1/20 0.43
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
POLB P06746 2/20 0.39
KDM4E B2RXH2 1/20 0.35
THRB P10828 1/20 0.34
LMNA P02545 2/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPT P10636 2/20 0.33
GRIA2 P42262 5/20 0.33
GRIA1 P42261 4/20 0.33
GRIA3 P42263 4/20 0.33
GRIA4 P48058 4/20 0.33
PER2 O15055 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5349703 0.88 NPSR1 (0.50) NPSR1TP53KMT2AMEN1POLB
SCHEMBL5358632 0.82 NPSR1 (0.40) NPSR1TP53KMT2AMEN1POLB
SCHEMBL5369657 0.78 NPSR1 (0.36) NPSR1TP53KMT2AMEN1POLB
SCHEMBL5361851 0.75 GRIA2 (0.48) NPSR1TP53KMT2AMEN1POLB
SCHEMBL5359272 0.75 NPSR1 (0.40) NPSR1TP53KMT2AMEN1POLB
SCHEMBL5354922 0.73 NPSR1 (0.34) NPSR1KMT2AMEN1POLBKDM4E
SCHEMBL5487001 0.72 THRB (0.46) NPSR1TP53KMT2AMEN1KDM4E
SCHEMBL2778463 0.71 GRIA2 (0.42) NPSR1TP53KMT2AMEN1KDM4E
SCHEMBL5358401 0.70 NPSR1 (0.35) NPSR1TP53KMT2AMEN1POLB
SCHEMBL29437629 0.69 GRIA2 (0.45) NPSR1TP53KMT2AMEN1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7268129-B2 Fluorinated benzothiadiazine compounds LES LABORATOIRES SERVIER (FR) 2007-09-11 US disclosed
CN-1308317-C New fluorinated benzothiadiazine compounds, a process for their preparation and pharmaceutical compositions containing them SERVIER LAB (FR) 2007-04-04 CN disclosed
CN-1680343-A New fluorinated benzothiadiazine compounds, a process for their preparation and pharmaceutical compositions containing them SERVIER LAB (FR) 2005-10-12 CN disclosed
US-20050165008-A1 Fluorinated benzothiadiazine compounds LES LABORATORIES SERVIER (FR) 2005-07-28 US disclosed
EP-1557412-A1 Fluorinated benzothiadiazine derivatives and their use as AMPA receptor modulators Les Laboratoires Servier (FR) 2005-07-27 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050165008-A1 Fluorinated benzothiadiazine compounds GRM1, GRIN1, GRIK5 NPSR1 132/4885TP53 4216/4885KMT2A 930/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.