SCHEMBL5358762

SCHEMBL5358762

Cc1cc(-c2ccc(C#N)cc2)c(C)n1Cc1cc(C#N)n[nH]1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 3/20 0.40
CCNC P24863 1/20 0.38
CDK8 P49336 1/20 0.38
AR P10275 7/20 0.37
PIK3R1 P27986 2/20 0.36
PIK3CA P42336 2/20 0.36
LMNA P02545 2/20 0.36
MAPT P10636 2/20 0.36
KDM4E B2RXH2 1/20 0.36
MARK3 P27448 1/20 0.34
GSK3A P49840 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
NOTUM Q6P988 1/20 0.34
KLKB1 P03952 1/20 0.33
KLK1 P06870 1/20 0.33
CHEK1 O14757 1/20 0.33
KDM1A O60341 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5354656 0.86 AR (0.40) CYP11B2CCNCCDK8ARPIK3R1
SCHEMBL5357164 0.84 CYP11B2 (0.39) CYP11B2CCNCCDK8ARPIK3R1
SCHEMBL5368138 0.84 CYP11B2 (0.38) CYP11B2CCNCCDK8ARPIK3R1
SCHEMBL5365592 0.82 CYP11B2 (0.41) CYP11B2CCNCCDK8ARPIK3R1
SCHEMBL14347747 0.80 MAPT (0.39) CYP11B2ARLMNAMAPTKDM4E
SCHEMBL6889076 0.78 AR (0.51) CYP11B2CCNCCDK8ARPIK3R1
SCHEMBL5362436 0.76 CYP11B2 (0.40) CYP11B2CCNCCDK8ARPIK3R1
SCHEMBL5365214 0.76 CYP11B2 (0.43) CYP11B2CCNCCDK8ARLMNA
SCHEMBL5361962 0.75 MAPT (0.43) CYP11B2ARLMNAMAPTKDM4E
SCHEMBL13362142 0.75 CCNC (0.35) CYP11B2CCNCCDK8ARPIK3R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007145349-A2 SUBSTITUTED PYRROLE DERIVATIVES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-12-21 WO disclosed
WO-2007145349-A2 SUBSTITUTED PYRROLE DERIVATIVES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-12-21 WO disclosed