SCHEMBL5359277

SCHEMBL5359277

Cc1c(C#N)c(-c2ccc(C#N)cc2)c(C)n1Cc1cc(CO)[nH]n1

nearest known ligand 0.61

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AR P10275 10/20 0.61
CYP11B2 P19099 2/20 0.36
CCNC P24863 1/20 0.36
CDK8 P49336 1/20 0.36
CHEK1 O14757 1/20 0.34
GRIA2 P42262 1/20 0.34
GRIA4 P48058 1/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
DHODH Q02127 1/20 0.33
FNTA P49354 1/20 0.33
FNTB P49356 1/20 0.33
TNIK Q9UKE5 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5362087 0.88 AR (0.60) ARCYP11B2CCNCCDK8CHEK1
SCHEMBL5373726 0.82 AR (0.61) ARCCNCCDK8CHEK1GRIA2
SCHEMBL5361524 0.81 AR (0.54) ARCYP11B2CCNCCDK8CHEK1
SCHEMBL14348166 0.81 AR (0.50) ARCYP11B2CCNCCDK8CHEK1
SCHEMBL5362232 0.80 AR (0.61) ARCYP11B2CCNCCDK8GRIA2
SCHEMBL5359879 0.79 AR (0.52) ARFNTAFNTB
SCHEMBL14348310 0.78 AR (0.53) ARCCNCCDK8CHEK1GRIA2
SCHEMBL4919002 0.77 AR (0.70) ARCYP11B2FNTAFNTB
SCHEMBL5370036 0.77 AR (0.49) ARFNTAFNTB
SCHEMBL14347768 0.76 AR (0.57) ARCYP11B2CCNCCDK8GRIA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007145349-A2 SUBSTITUTED PYRROLE DERIVATIVES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-12-21 WO disclosed