SCHEMBL5362087

SCHEMBL5362087

Cc1cc(Cn2c(C)c(C#N)c(-c3ccc(C#N)cc3)c2C)n[nH]1

nearest known ligand 0.60

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AR P10275 10/20 0.60
CCNC P24863 1/20 0.41
CDK8 P49336 1/20 0.41
DHODH Q02127 1/20 0.39
CHEK1 O14757 1/20 0.37
CYP11B2 P19099 2/20 0.36
SLC11A2 P49281 1/20 0.36
KCNH2 Q12809 1/20 0.35
GRIN2B Q13224 1/20 0.35
GRIA2 P42262 1/20 0.34
GRIA4 P48058 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14348166 0.92 AR (0.50) ARCCNCCDK8DHODHCHEK1
SCHEMBL5359277 0.88 AR (0.61) ARCCNCCDK8DHODHCHEK1
SCHEMBL5361524 0.85 AR (0.54) ARCCNCCDK8CHEK1CYP11B2
SCHEMBL5373726 0.84 AR (0.61) ARCCNCCDK8CHEK1GRIA2
SCHEMBL5362232 0.84 AR (0.61) ARCCNCCDK8DHODHCYP11B2
SCHEMBL5359879 0.81 AR (0.52) AR
SCHEMBL6469428 0.79 AR (0.58) ARCCNCCDK8CYP11B2SLC11A2
SCHEMBL6466733 0.79 AR (0.60) ARCYP11B2SLC11A2GRIA2GRIA4
SCHEMBL6468889 0.78 AR (0.86) ARCCNCCDK8CYP11B2
SCHEMBL14348310 0.78 AR (0.53) ARCCNCCDK8CHEK1GRIA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007145349-A2 SUBSTITUTED PYRROLE DERIVATIVES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-12-21 WO disclosed