SCHEMBL5361772

SCHEMBL5361772

Cc1c(C#N)c(-c2ccc(C#N)cc2)c(C)n1Cc1csc(C(F)(F)F)n1

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AR P10275 8/20 0.53
GAA P10253 1/20 0.37
CYP11B2 P19099 3/20 0.36
CNR1 P21554 4/20 0.35
RIPK3 Q9Y572 1/20 0.34
KIF11 P52732 1/20 0.33
GRIA2 P42262 1/20 0.33
GRIA4 P48058 1/20 0.33
SDHB P21912 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5360218 0.83 AR (0.53) ARGAACYP11B2CNR1SDHB
SCHEMBL5366353 0.77 AR (0.60) ARCYP11B2GRIA2GRIA4
SCHEMBL5361524 0.77 AR (0.54) ARCYP11B2KIF11
SCHEMBL5362024 0.76 AR (0.58) ARGAACYP11B2GRIA2GRIA4
SCHEMBL5365976 0.75 AR (0.52) ARGAACYP11B2GRIA2GRIA4
SCHEMBL5362158 0.75 AR (0.53) ARCYP11B2CNR1
SCHEMBL6466987 0.74 AR (0.58) ARCYP11B2GRIA2GRIA4
SCHEMBL6466733 0.74 AR (0.60) ARCYP11B2GRIA2GRIA4
SCHEMBL14347633 0.74 AR (0.58) ARGAACYP11B2GRIA2GRIA4
SCHEMBL5362232 0.73 AR (0.61) ARCYP11B2GRIA2GRIA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007145349-A2 SUBSTITUTED PYRROLE DERIVATIVES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-12-21 WO disclosed
WO-2007145349-A2 SUBSTITUTED PYRROLE DERIVATIVES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-12-21 WO disclosed