SCHEMBL5365976

SCHEMBL5365976

Cc1c(C#N)c(-c2ccc(C#N)cc2)c(C)n1Cc1nc(C(C)(C)O)cs1

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AR P10275 10/20 0.52
GAA P10253 1/20 0.36
MAPK1 P28482 1/20 0.36
GRIA2 P42262 1/20 0.32
GRIA4 P48058 1/20 0.32
CYP11B2 P19099 2/20 0.32
KDM4E B2RXH2 1/20 0.32
LMNA P02545 1/20 0.32
MAPT P10636 1/20 0.32
KDM1A O60341 1/20 0.32
FNTA P49354 1/20 0.31
FNTB P49356 1/20 0.31
SLC22A12 Q96S37 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5360218 0.88 AR (0.53) ARGAAMAPK1CYP11B2
SCHEMBL6464529 0.77 AR (0.69) ARCYP11B2KDM1A
SCHEMBL5361772 0.75 AR (0.53) ARGAAGRIA2GRIA4CYP11B2
SCHEMBL5365843 0.75 AR (0.58) ARGAACYP11B2LMNAMAPT
SCHEMBL14347707 0.74 AR (0.58) ARGRIA2GRIA4CYP11B2FNTA
SCHEMBL6464438 0.72 AR (0.73) ARCYP11B2KDM1ASLC22A12
SCHEMBL5367267 0.72 AR (0.52) ARGRIA2GRIA4CYP11B2KDM1A
SCHEMBL5362158 0.72 AR (0.53) ARCYP11B2FNTAFNTB
SCHEMBL6468889 0.72 AR (0.86) ARCYP11B2KDM4E
SCHEMBL14347629 0.71 AR (0.43) ARMAPK1GRIA2GRIA4KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007145349-A2 SUBSTITUTED PYRROLE DERIVATIVES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-12-21 WO disclosed