SCHEMBL5366353

SCHEMBL5366353

Cc1c(C#N)c(-c2ccc(C#N)cc2)c(C)n1Cc1ccn(C)n1

nearest known ligand 0.60

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
AR P10275 8/20 0.60
CYP11B2 P19099 2/20 0.38
KDM1A O60341 1/20 0.36
GRIA2 P42262 2/20 0.36
GRIA4 P48058 2/20 0.36
KCNH2 Q12809 6/20 0.36
GRIN2B Q13224 1/20 0.36
ADORA2B P29275 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14348165 0.90 AR (0.48) ARCYP11B2KDM1AGRIA2GRIA4
SCHEMBL5369671 0.80 AR (0.60) ARCYP11B2GRIA2GRIA4
SCHEMBL6466733 0.79 AR (0.60) ARCYP11B2GRIA2GRIA4
SCHEMBL6466987 0.79 AR (0.58) ARCYP11B2GRIA2GRIA4
SCHEMBL5362232 0.79 AR (0.61) ARCYP11B2GRIA2GRIA4
SCHEMBL6468889 0.78 AR (0.86) ARCYP11B2
SCHEMBL5362087 0.78 AR (0.60) ARCYP11B2GRIA2GRIA4KCNH2
SCHEMBL6466150 0.78 AR (0.69) ARCYP11B2GRIN2B
SCHEMBL5361772 0.77 AR (0.53) ARCYP11B2GRIA2GRIA4
SCHEMBL5365931 0.77 AR (0.65) ARCYP11B2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007145349-A2 SUBSTITUTED PYRROLE DERIVATIVES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-12-21 WO disclosed