SCHEMBL536230

SCHEMBL536230

CCc1ccccc1-c1ccc(C(=O)O)cc1C(F)(F)F.Cc1ccccc1-c1ccc(C(=O)O)cc1C

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
RORC P51449 2/20 0.42
GPBAR1 Q8TDU6 4/20 0.42
AKR1C3 P42330 3/20 0.42
AKR1C2 P52895 3/20 0.42
RARB P10826 1/20 0.41
PPARD Q03181 2/20 0.40
SRD5A2 P31213 1/20 0.40
ADH5 P11766 1/20 0.40
S1PR1 P21453 1/20 0.40
PTPRC P08575 2/20 0.40
EPHX2 P34913 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL410339 0.91 AKR1C3 (0.47) GPBAR1AKR1C3AKR1C2SRD5A2ADH5
SCHEMBL319595 0.89 GPBAR1 (0.49) RORCGPBAR1AKR1C3AKR1C2RARB
SCHEMBL319915 0.83 RORC (0.52) RORCAKR1C3AKR1C2SRD5A2S1PR1
SCHEMBL272092 0.79 TTR (0.56) SRD5A2PTPRC
SCHEMBL536675 0.78 NOTUM (0.51) AKR1C3AKR1C2
SCHEMBL272324 0.77 PTPRC (0.54) AKR1C3AKR1C2SRD5A2ADH5PTPRC
SCHEMBL336261 0.76 ADH5 (0.54) AKR1C3AKR1C2RARBSRD5A2ADH5
SCHEMBL320542 0.75 NOTUM (0.54) GPBAR1AKR1C3AKR1C2S1PR1
SCHEMBL13601649 0.75 RORC (0.49) RORCGPBAR1AKR1C3AKR1C2RARB
SCHEMBL13601671 0.75 RORC (0.47) RORCAKR1C3AKR1C2RARBSRD5A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2414342-A1 OXADIAZOLE DERIVATIVES Merck Serono S.A. (CH) 2012-02-08 EP disclosed
WO-2010112461-A1 OXADIAZOLE DERIVATIVES MERCK SERONO S.A. (CH) 2010-10-07 WO disclosed