SCHEMBL5362350

SCHEMBL5362350

Cc1c(C#N)c(-c2ccc(C#N)cc2)c(C)n1Cc1nc(C#N)co1

nearest known ligand 0.57

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AR P10275 10/20 0.57
CYP11B2 P19099 3/20 0.35
GRIA2 P42262 1/20 0.33
GRIA4 P48058 1/20 0.33
GHSR Q92847 1/20 0.32
GAA P10253 1/20 0.32
CRHR1 P34998 1/20 0.32
PDE9A O76083 1/20 0.32
PDE1C Q14123 1/20 0.32
CYP11B1 P15538 1/20 0.32
PTPN11 Q06124 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5366328 0.83 AR (0.60) ARGRIA2GRIA4
SCHEMBL14348320 0.82 AR (0.53) ARGRIA2GRIA4
SCHEMBL5358252 0.81 AR (0.52) ARCYP11B2GRIA2GRIA4CYP11B1
SCHEMBL6468079 0.80 AR (0.58) ARCYP11B2
SCHEMBL14347633 0.80 AR (0.58) ARCYP11B2GRIA2GRIA4GAA
SCHEMBL6468889 0.76 AR (0.86) ARCYP11B2PDE9APDE1CCYP11B1
SCHEMBL5361589 0.75 AR (0.61) ARCYP11B2GRIA2GRIA4CYP11B1
SCHEMBL5357480 0.74 AR (0.61) ARCYP11B2GRIA2GRIA4
SCHEMBL6465872 0.74 AR (0.76) ARCYP11B2PDE9APDE1CCYP11B1
SCHEMBL24414502 0.73 AR (0.80) ARCYP11B2PDE9APDE1CCYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007145349-A2 SUBSTITUTED PYRROLE DERIVATIVES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-12-21 WO claimed
WO-2007145349-A2 SUBSTITUTED PYRROLE DERIVATIVES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-12-21 WO disclosed