SCHEMBL5364856

SCHEMBL5364856

O=c1ccc(Cc2ccc(Cl)c(Oc3cccc(Br)c3)c2F)n[nH]1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 6/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
THRA P10827 2/20 0.41
THRB P10828 2/20 0.41
AKR1B1 P15121 6/20 0.36
SOD1 P00441 1/20 0.33
GRM4 Q14833 1/20 0.32
NPBWR1 P48145 1/20 0.31
HTR2A P28223 1/20 0.31
SLC6A4 P31645 1/20 0.31
KCNH2 Q12809 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5377018 0.90 THRA (0.44) CYP3A4CYP2C9CYP2C19THRATHRB
SCHEMBL5373738 0.88 CYP3A4 (0.41) CYP3A4CYP2C9CYP2C19THRATHRB
SCHEMBL5367059 0.87 CYP3A4 (0.48) CYP3A4CYP2C9CYP2C19THRATHRB
SCHEMBL5365045 0.85 CYP3A4 (0.44) CYP3A4CYP2C9CYP2C19THRATHRB
SCHEMBL14570716 0.85 CYP3A4 (0.60) CYP3A4CYP2C9CYP2C19THRATHRB
SCHEMBL5377753 0.83 CYP3A4 (0.45) CYP3A4CYP2C9CYP2C19THRATHRB
SCHEMBL5364622 0.80 CYP3A4 (0.43) CYP3A4CYP2C9CYP2C19THRATHRB
SCHEMBL5368884 0.80 CYP3A4 (0.68) CYP3A4CYP2C9CYP2C19THRATHRB
SCHEMBL5373847 0.78 THRA (0.44) CYP3A4CYP2C9CYP2C19THRATHRB
SCHEMBL5368441 0.78 CYP3A4 (0.58) CYP3A4CYP2C9CYP2C19THRATHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed