SCHEMBL5365095

SCHEMBL5365095

Cc1c(C#N)c(-c2ccc(C#N)cc2)c(C)n1Cc1cnn(C(c2ccccc2)(c2ccccc2)c2ccccc2)c1

nearest known ligand 0.65

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AR P10275 11/20 0.65
PDE9A O76083 1/20 0.36
PDE1C Q14123 1/20 0.36
CYP11B2 P19099 4/20 0.36
CYP11B1 P15538 2/20 0.33
GRIA2 P42262 1/20 0.33
GRIA4 P48058 1/20 0.33
CYP19A1 P11511 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
PKM P14618 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6525379 0.82 AR (0.58) ARGRIA2GRIA4CYP19A1
SCHEMBL5369671 0.80 AR (0.60) ARPDE9APDE1CCYP11B2GRIA2
SCHEMBL5365931 0.80 AR (0.65) ARCYP11B2CYP11B1
SCHEMBL5358573 0.79 AR (0.54) ARGRIA2GRIA4ALDH1A1
SCHEMBL6466386 0.78 AR (0.58) ARGRIA2GRIA4CYP19A1
SCHEMBL6468889 0.76 AR (0.86) ARPDE9APDE1CCYP11B2CYP11B1
SCHEMBL6466161 0.76 AR (0.58) ARPDE9APDE1CGRIA2GRIA4
SCHEMBL6465272 0.74 AR (1.00) ARPDE9APDE1CCYP11B2CYP11B1
SCHEMBL6464451 0.73 AR (0.80) ARCYP11B2CYP11B1CYP19A1
SCHEMBL6465872 0.73 AR (0.76) ARPDE9APDE1CCYP11B2CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007145349-A2 SUBSTITUTED PYRROLE DERIVATIVES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-12-21 WO disclosed