SCHEMBL5358573

SCHEMBL5358573

Cc1c(C#N)c(-c2ccc(C#N)cc2)c(C)n1Cc1cn(C(c2ccccc2)(c2ccccc2)c2ccccc2)nc1C(F)(F)F

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 10/20 0.54
PPARD Q03181 1/20 0.34
SLC2A1 P11166 3/20 0.33
SLC2A3 P11169 3/20 0.33
SLC2A4 P14672 3/20 0.33
CNR1 P21554 1/20 0.32
KIF11 P52732 1/20 0.32
SLC2A2 P11168 1/20 0.32
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
MAPT P10636 1/20 0.31
HTT P42858 1/20 0.31
NCOA1 Q15788 1/20 0.31
NCOA3 Q9Y6Q9 1/20 0.31
GRIA2 P42262 1/20 0.31
GRIA4 P48058 1/20 0.31
GABRP O00591 1/20 0.31
GABRD O14764 1/20 0.31
GABRA1 P14867 1/20 0.31
GABRB1 P18505 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5369671 0.79 AR (0.60) ARLMNAMAPTGRIA2GRIA4
SCHEMBL6525379 0.79 AR (0.58) ARGRIA2GRIA4
SCHEMBL5365095 0.79 AR (0.65) ARALDH1A1GRIA2GRIA4
SCHEMBL14347772 0.75 AR (0.53) ARPPARDCNR1KIF11
SCHEMBL6466386 0.75 AR (0.58) ARGRIA2GRIA4
SCHEMBL5362174 0.74 AR (0.44) ARKIF11
SCHEMBL6466161 0.73 AR (0.58) ARALDH1A1GRIA2GRIA4
SCHEMBL5362158 0.70 AR (0.53) ARSLC2A1SLC2A3SLC2A4CNR1
SCHEMBL5358210 0.70 AR (0.47) AR
SCHEMBL24112327 0.69 ALDH1A1 (0.34) ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007145349-A2 SUBSTITUTED PYRROLE DERIVATIVES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-12-21 WO disclosed