SCHEMBL5369671

SCHEMBL5369671

Cc1c(C#N)c(-c2ccc(C#N)cc2)c(C)n1Cc1ccn(C(c2ccccc2)(c2ccccc2)c2ccccc2)n1

nearest known ligand 0.60

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AR P10275 8/20 0.60
GRIA2 P42262 2/20 0.34
GRIA4 P48058 2/20 0.34
PDE9A O76083 1/20 0.33
PDE1C Q14123 1/20 0.33
ACSS2 Q9NR19 1/20 0.32
CYP11B2 P19099 1/20 0.32
KDM4E B2RXH2 1/20 0.32
MAPT P10636 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
SLC11A2 P49281 1/20 0.31
LMNA P02545 1/20 0.31
TSHR P16473 1/20 0.31
NTRK1 P04629 1/20 0.31
NTRK3 Q16288 1/20 0.31
NTRK2 Q16620 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6525379 0.84 AR (0.58) ARGRIA2GRIA4
SCHEMBL5365095 0.80 AR (0.65) ARGRIA2GRIA4PDE9APDE1C
SCHEMBL6466386 0.80 AR (0.58) ARGRIA2GRIA4SLC11A2
SCHEMBL5366353 0.80 AR (0.60) ARGRIA2GRIA4CYP11B2
SCHEMBL5358573 0.79 AR (0.54) ARGRIA2GRIA4MAPTLMNA
SCHEMBL6466161 0.78 AR (0.58) ARGRIA2GRIA4PDE9APDE1C
SCHEMBL5358210 0.76 AR (0.47) ARACSS2
SCHEMBL5362174 0.73 AR (0.44) AR
SCHEMBL5362232 0.72 AR (0.61) ARGRIA2GRIA4CYP11B2KDM4E
SCHEMBL6468889 0.71 AR (0.86) ARPDE9APDE1CCYP11B2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007145349-A2 SUBSTITUTED PYRROLE DERIVATIVES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-12-21 WO disclosed