SCHEMBL5367267

SCHEMBL5367267

Cc1c(C#N)c(-c2ccc(C#N)cc2)c(C)n1Cc1c[nH]nc1C(C)(C)O

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AR P10275 10/20 0.52
KDM1A O60341 1/20 0.33
GRIA2 P42262 1/20 0.32
GRIA4 P48058 1/20 0.32
FNTA P49354 5/20 0.32
FNTB P49356 5/20 0.32
CYP11B2 P19099 2/20 0.32
CCNC P24863 1/20 0.31
CDK8 P49336 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14347772 0.88 AR (0.53) ARCYP11B2CCNCCDK8
SCHEMBL14347768 0.83 AR (0.57) ARKDM1AGRIA2GRIA4FNTA
SCHEMBL5357688 0.82 CYP11B2 (0.36) ARKDM1AFNTAFNTBCYP11B2
SCHEMBL5362254 0.81 AR (0.60) ARGRIA2GRIA4FNTAFNTB
SCHEMBL14348167 0.80 AR (0.53) ARGRIA2GRIA4FNTAFNTB
SCHEMBL5368784 0.78 AR (0.58) ARGRIA2GRIA4FNTAFNTB
SCHEMBL5362232 0.75 AR (0.61) ARGRIA2GRIA4FNTAFNTB
SCHEMBL6464438 0.74 AR (0.73) ARKDM1ACYP11B2
SCHEMBL6464529 0.73 AR (0.69) ARKDM1ACYP11B2
SCHEMBL6469428 0.73 AR (0.58) ARGRIA2GRIA4FNTAFNTB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007145349-A2 SUBSTITUTED PYRROLE DERIVATIVES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-12-21 WO disclosed
WO-2007145349-A2 SUBSTITUTED PYRROLE DERIVATIVES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-12-21 WO disclosed