SCHEMBL5366358

SCHEMBL5366358

NCCCCC(N)(CCCN)CCCN

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFKB1 P19838 2/20 0.47
DNM1 Q05193 3/20 0.44
CA12 O43570 2/20 0.44
CA1 P00915 2/20 0.44
CA2 P00918 2/20 0.44
CA3 P07451 2/20 0.44
CA4 P22748 2/20 0.44
CA6 P23280 2/20 0.44
CA5A P35218 2/20 0.44
CA7 P43166 2/20 0.44
CA9 Q16790 2/20 0.44
CA14 Q9ULX7 2/20 0.44
CA5B Q9Y2D0 2/20 0.44
BLM P54132 2/20 0.44
LMNA P02545 1/20 0.44
TSHR P16473 1/20 0.44
FDPS P14324 3/20 0.39
ODC1 P11926 2/20 0.36
CYP2D6 P10635 1/20 0.35
PDE3A Q14432 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2357721 1.00 NFKB1 (0.47) NFKB1DNM1CA12CA1CA2
SCHEMBL817872 0.97 DNM1 (0.50) NFKB1DNM1CA12CA1CA2
SCHEMBL7093120 0.97 DNM1 (0.50) NFKB1DNM1CA12CA1CA2
SCHEMBL28300322 0.97 DNM1 (0.50) NFKB1DNM1CA12CA1CA2
SCHEMBL20425510 0.93 DNM1 (0.53) NFKB1DNM1CA12CA1CA2
SCHEMBL816414 0.93 NFKB1 (0.43) NFKB1DNM1CA12CA1CA2
Water SCHEMBL30354056 0.90 NFKB1 (0.40) NFKB1DNM1CA12CA1CA2
Hydrochloric Acid SCHEMBL16398251 0.90 NFKB1 (0.40) NFKB1DNM1CA12CA1CA2
SCHEMBL3128429 0.89 NFKB1 (0.37) NFKB1DNM1CA12CA1CA2
SCHEMBL817593 0.88 DNM1 (0.47) NFKB1DNM1CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001927-A2 NOVEL POLYAMINE ANALOGUES AS THERAPEUTIC AND DIAGNOSTIC AGENTS ORIDIGM CORPORATION (US) 2000-05-24 EP claimed
WO-1999003823-A2 NOVEL POLYAMINE ANALOGUES AS THERAPEUTIC AND DIAGNOSTIC AGENTS ORIDIGM CORPORATION (US) 1999-01-28 WO claimed
CN-102686222-B Orally delivered drugs comprising MGBG and methods of treating diseases PATHOLOGICA LLC 2015-06-24 CN disclosed
EP-1867633-A1 Polyamine analogues as therapeutic and diagnostic agents MediQuest Therapeutics, Inc. (US) 2007-12-19 EP disclosed
US-7208528-B1 Polyamine analogues as therapeutic and diagnostic agents MEDIQUEST THERAPEUTICS, INC. (US) 2007-04-24 US disclosed
US-7160923-B1 Polyamine analogues as therapeutic and diagnostic agents MEDIQUEST THERAPEUTICS, INC. (US) 2007-01-09 US disclosed
EP-1317424-A2 POLYAMINE ANALOGUES AS THERAPEUTIC AND DIAGNOSTIC AGENTS MediQuest Therapeutics, Inc. (US) 2003-06-11 EP disclosed
WO-2001092218-A2 POLYAMINE ANALOGUES AS THERAPEUTIC AND DIAGNOSTIC AGENTS ORIDIGM CORPORATION (US) 2001-12-06 WO disclosed
EP-1085011-A1 Novel polyamine analogues as therapeutic and diagnostic agents ORIDIGM CORPORATION (US) 2001-03-21 EP disclosed
US-6172261-B1 BIOSYNTHESIS USING CHAIN EXTENSION ORIDIGM CORPORATION 2001-01-09 US disclosed
EP-1001927-A2 NOVEL POLYAMINE ANALOGUES AS THERAPEUTIC AND DIAGNOSTIC AGENTS ORIDIGM CORPORATION (US) 2000-05-24 EP disclosed
WO-1999003823-A2 NOVEL POLYAMINE ANALOGUES AS THERAPEUTIC AND DIAGNOSTIC AGENTS ORIDIGM CORPORATION (US) 1999-01-28 WO disclosed