SCHEMBL5366565

SCHEMBL5366565

COC(=O)C=C[C@H](Cc1ccc(OCc2ccccc2)cc1)NC(=O)OC(C)(C)C

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 4/20 0.53
BCL2 P10415 1/20 0.52
YAP1 P46937 3/20 0.49
PPARG P37231 3/20 0.49
CTSL P07711 1/20 0.48
HDAC8 Q9BY41 1/20 0.48
PPARA Q07869 1/20 0.47
REN P00797 1/20 0.47
ITGB3 P05106 1/20 0.47
ITGA2B P08514 1/20 0.47
LTA4H P09960 1/20 0.47
ATM Q13315 1/20 0.45
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5356751 1.00 PTPN1 (0.53) PTPN1BCL2YAP1PPARGCTSL
SCHEMBL5356760 1.00 PTPN1 (0.53) PTPN1BCL2YAP1PPARGCTSL
SCHEMBL5356756 1.00 PTPN1 (0.53) PTPN1BCL2YAP1PPARGCTSL
SCHEMBL21214703 0.91 PTPN1 (0.51) PTPN1BCL2YAP1PPARGCTSL
SCHEMBL5358030 0.91 PTPN1 (0.51) PTPN1BCL2YAP1PPARGCTSL
SCHEMBL5358032 0.91 PTPN1 (0.51) PTPN1BCL2YAP1PPARGCTSL
SCHEMBL5406758 0.90 ATM (0.53) PPARGCTSLPPARARENATM
SCHEMBL5406769 0.90 ATM (0.53) PPARGCTSLPPARARENATM
SCHEMBL5416888 0.90 ATM (0.53) PPARGCTSLPPARARENATM
SCHEMBL5406765 0.90 ATM (0.53) PPARGCTSLPPARARENATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7253194-B2 Compounds and inhibitors of phospholipases THE UNIVERSITY OF QUEENSLAND (AU) 2007-08-07 US disclosed
EP-1309552-A4 COMPOUNDS AND INHIBITORS OF PHOSPHOLIPASES UNIV QUEENSLAND (AU) 2005-07-20 EP disclosed
US-20040033995-A1 Compounds and inhibitors of phospholipases QUEENSLAND, THE UNIVERSITY OF (AU) 2004-02-19 US disclosed
EP-1309552-A1 COMPOUNDS AND INHIBITORS OF PHOSPHOLIPASES THE UNIVERSITY OF QUEENSLAND (AU) 2003-05-14 EP disclosed
WO-2002008189-A1 COMPOUNDS AND INHIBITORS OF PHOSPHOLIPASES THE UNIVERSITY OF QUEENSLAND (AU) 2002-01-31 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040033995-A1 Compounds and inhibitors of phospholipases PLA2G4C, PLA2G4B, PLA2G4A PTPN1 1814/4885BCL2 2789/4885YAP1 4254/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.