SCHEMBL5366963

SCHEMBL5366963

Cc1cc(=O)[nH]nc1Cc1ccc(Cl)c(Oc2cc(C#N)cc(C(F)F)c2)c1F

nearest known ligand 0.58

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.58
CYP2C9 P11712 1/20 0.58
CYP2C19 P33261 1/20 0.58
KCNH2 Q12809 5/20 0.38
RORC P51449 1/20 0.33
EPAS1 Q99814 2/20 0.32
HTR2A P28223 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5331103 0.85 CYP3A4 (0.61) CYP3A4CYP2C9CYP2C19KCNH2RORC
SCHEMBL5344677 0.85 CYP3A4 (0.81) CYP3A4CYP2C9CYP2C19KCNH2RORC
SCHEMBL4810352 0.83 CYP3A4 (0.68) CYP3A4CYP2C9CYP2C19KCNH2RORC
SCHEMBL1341943 0.81 CYP3A4 (0.47) CYP3A4CYP2C9CYP2C19KCNH2RORC
SCHEMBL13492117 0.81 CYP3A4 (0.50) CYP3A4CYP2C9CYP2C19KCNH2RORC
SCHEMBL1344843 0.80 CYP3A4 (0.47) CYP3A4CYP2C9CYP2C19KCNH2RORC
SCHEMBL1343995 0.80 CYP3A4 (0.47) CYP3A4CYP2C9CYP2C19KCNH2RORC
SCHEMBL11904766 0.78 CYP3A4 (0.51) CYP3A4CYP2C9CYP2C19KCNH2RORC
SCHEMBL4370334 0.77 CYP3A4 (0.61) CYP3A4CYP2C9CYP2C19RORCEPAS1
SCHEMBL4368132 0.77 CYP3A4 (0.61) CYP3A4CYP2C9CYP2C19RORCEPAS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed