SCHEMBL5368026

SCHEMBL5368026

Nc1c(Br)cc(C(=O)NCC(=O)N2CCC(n3c(=O)[nH]c4ccccc43)CC2)cc1Br

nearest known ligand 0.55

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PLD2 O14939 16/20 0.55
PLD1 Q13393 13/20 0.55
HSD11B1 P28845 2/20 0.51
ALDH1A1 P00352 1/20 0.50
MAPK1 P28482 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5377748 0.91 PLD2 (0.58) PLD2PLD1
SCHEMBL5366246 0.85 PLD2 (0.76) PLD2PLD1
SCHEMBL5367571 0.85 HSD11B1 (0.52) HSD11B1ALDH1A1MAPK1
SCHEMBL5365941 0.82 HSD11B1 (0.52) HSD11B1
SCHEMBL5369875 0.79 CALCRL (0.48)
SCHEMBL3960728 0.78 CALCRL (0.71) ALDH1A1MAPK1
SCHEMBL5372045 0.78 HSD11B1 (0.57) HSD11B1ALDH1A1MAPK1
SCHEMBL5369487 0.77 CHRM1 (0.70) PLD2PLD1ALDH1A1MAPK1
Hydrochloric Acid SCHEMBL5366218 0.76 CHRM1 (0.69) PLD2PLD1ALDH1A1MAPK1
SCHEMBL3960471 0.76 CALCRL (0.69)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7230001-B1 Arylalkane, arylalkene and aryl azaalkane, medicaments containing said compounds and method for the production thereof BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2007-06-12 US disclosed