SCHEMBL5368386

SCHEMBL5368386

Cc1ccc(CCS(=O)(=O)N2CCC(CNC(=O)c3ccncc3)CC2)cc1

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
F10 P00742 6/20 0.51
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
HDAC6 Q9UBN7 1/20 0.49
KCNH2 Q12809 1/20 0.48
CACNA1I Q9P0X4 1/20 0.48
ALDH1A1 P00352 3/20 0.48
HPGD P15428 1/20 0.48
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
MMP13 P45452 1/20 0.43
USP30 Q70CQ3 1/20 0.43
NAMPT P43490 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5368614 0.90 HDAC6 (0.55) HDAC6RAB9AUSP30
SCHEMBL14425183 0.86 MEN1 (0.47) F10MEN1KMT2AHDAC6KCNH2
SCHEMBL14425189 0.85 MEN1 (0.48) F10MEN1KMT2AHDAC6KCNH2
SCHEMBL14425186 0.79 HDAC6 (0.51) F10HDAC6CACNA1IALDH1A1SMN1; SMN2
SCHEMBL5366612 0.78 HDAC6 (0.52) F10MEN1KMT2AHDAC6ALDH1A1
SCHEMBL5368330 0.78 HDAC6 (0.52) F10HDAC6KCNH2CACNA1INPC1
SCHEMBL14425184 0.78 HDAC6 (0.52) F10HDAC6CACNA1IALDH1A1SMN1; SMN2
SCHEMBL5362714 0.78 HDAC6 (0.59) HDAC6
SCHEMBL5350879 0.77 GRIN2B (0.57) MEN1KMT2AHDAC6ALDH1A1HPGD
SCHEMBL5374920 0.76 TPSAB1 (0.66) F10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed