SCHEMBL5368330

SCHEMBL5368330

O=C(NCC1CCN(S(=O)(=O)CCc2ccc(Cl)cc2)CC1)c1ccc(O)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 3/20 0.52
SMN1; SMN2 Q16637 2/20 0.52
GAA P10253 2/20 0.52
MAPT P10636 2/20 0.52
NPC1 O15118 1/20 0.52
CYP1A2 P05177 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C19 P33261 1/20 0.52
RAB9A P51151 1/20 0.52
GFER P55789 1/20 0.52
LMNA P02545 2/20 0.52
KDM4E B2RXH2 1/20 0.52
HTT P42858 1/20 0.52
CXCR3 P49682 3/20 0.48
TGM2 P21980 1/20 0.48
CCR2 P41597 2/20 0.48
HDAC3 O15379 2/20 0.46
HDAC4 P56524 2/20 0.46
HDAC1 Q13547 2/20 0.46
HDAC7 Q8WUI4 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5366612 0.90 HDAC6 (0.52) HDAC6SMN1; SMN2GAARAB9ALMNA
SCHEMBL5362714 0.89 HDAC6 (0.59) HDAC6CYP2C19LMNATGM2HDAC3
SCHEMBL5368040 0.81 CCR2 (0.69) HDAC6CCR2HDAC3HDAC4HDAC1
SCHEMBL5359321 0.80 HDAC6 (0.47) HDAC6KDM4ECXCR3HDAC3HDAC4
SCHEMBL5368386 0.78 F10 (0.51) HDAC6SMN1; SMN2NPC1RAB9AF10
SCHEMBL5368614 0.78 HDAC6 (0.55) HDAC6CYP2C19RAB9ALMNAHDAC3
SCHEMBL5363063 0.77 HDAC6 (0.52) HDAC6SMN1; SMN2MAPTNPC1CYP2C19
SCHEMBL5366291 0.77 TPSAB1 (0.72) SMN1; SMN2GAAMAPTNPC1CYP1A2
SCHEMBL14425184 0.75 HDAC6 (0.52) HDAC6SMN1; SMN2CYP2C19LMNAHDAC3
SCHEMBL14425189 0.74 MEN1 (0.48) HDAC6LMNAF10KCNH2CACNA1I

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed