SCHEMBL5368583

SCHEMBL5368583

Cc1cc(C(=O)NCC2CN(CCc3ccccc3)CCO2)ccc1O

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.48
HPGD P15428 3/20 0.48
KDM4E B2RXH2 2/20 0.48
ALDH1A1 P00352 2/20 0.48
GAA P10253 2/20 0.48
HSD17B10 Q99714 1/20 0.48
CACNA1H O95180 1/20 0.47
DRD4 P21917 4/20 0.44
DRD2 P14416 1/20 0.44
DRD3 P35462 1/20 0.44
POLB P06746 2/20 0.43
RAB9A P51151 1/20 0.42
ESRRG P62508 1/20 0.42
HTR1A P08908 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5360946 0.90 EPHX2 (0.47) EPHX2HPGDKDM4EALDH1A1GAA
SCHEMBL5366013 0.87 DRD4 (0.56) EPHX2HPGDKDM4EALDH1A1GAA
SCHEMBL14425319 0.87 DRD4 (0.56) EPHX2HPGDKDM4EALDH1A1GAA
SCHEMBL18487141 0.87 HPGD (0.55) EPHX2HPGDKDM4EALDH1A1GAA
SCHEMBL5360176 0.83 HPGD (0.45) EPHX2HPGDKDM4EALDH1A1GAA
SCHEMBL5365324 0.82 CCR3 (0.49) EPHX2HPGDKDM4EALDH1A1GAA
SCHEMBL5368664 0.81 DRD4 (0.54) EPHX2HPGDKDM4EALDH1A1GAA
SCHEMBL5366509 0.81 SMN1; SMN2 (0.58) EPHX2HPGDKDM4EALDH1A1GAA
SCHEMBL14425328 0.81 KDM4E (0.53) EPHX2HPGDKDM4EALDH1A1GAA
SCHEMBL5374908 0.80 ENPP2 (0.48) EPHX2HPGDPOLBRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed