SCHEMBL5368728

SCHEMBL5368728

CNS(=O)(=O)c1ccc2c(c1)C(=Cc1cc(Cl)cc(Br)c1O)C(=O)N2

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 4/20 0.53
PSEN1 P49768 1/20 0.53
PSEN2 P49810 1/20 0.53
APH1B Q8WW43 1/20 0.53
NCSTN Q92542 1/20 0.53
APH1A Q96BI3 1/20 0.53
PSENEN Q9NZ42 1/20 0.53
SRC P12931 3/20 0.51
NTRK1 P04629 3/20 0.51
FCER2 P06734 1/20 0.51
SYK P43405 1/20 0.51
NTRK3 Q16288 1/20 0.51
NTRK2 Q16620 1/20 0.51
CDK2 P24941 2/20 0.49
RAF1 P04049 5/20 0.48
KDR P35968 2/20 0.48
MDM2 Q00987 1/20 0.47
AURKA O14965 2/20 0.46
LCK P06239 1/20 0.45
FYN P06241 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5367143 0.90 SRC (0.52) LRRK2PSEN1PSEN2APH1BNCSTN
SCHEMBL5366300 0.90 SRC (0.52) LRRK2PSEN1PSEN2APH1BNCSTN
SCHEMBL5358785 0.87 SYK (0.61) LRRK2SRCNTRK1FCER2SYK
SCHEMBL5365765 0.85 SRC (0.52) LRRK2PSEN1PSEN2APH1BNCSTN
SCHEMBL5358529 0.82 MOGAT2 (0.51) LRRK2PSEN1PSEN2APH1BNCSTN
SCHEMBL5364961 0.82 MAP1LC3B (0.67) LRRK2PSEN1PSEN2APH1BNCSTN
SCHEMBL5365553 0.81 PLK4 (0.53) SRCNTRK1FCER2SYKNTRK3
SCHEMBL7137047 0.81 SRC (0.52) LRRK2PSEN1PSEN2APH1BNCSTN
SCHEMBL7139608 0.81 SRC (0.54) LRRK2SRCNTRK1FCER2SYK
SCHEMBL5360933 0.81 MAP3K7 (0.58) SRCNTRK1FCER2SYKNTRK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7202265-B2 Indolinone combinatorial libraries and related products and methods for the treatment of disease SUGEN, INC. (US) 2007-04-10 US disclosed
US-20050197382-A1 Indolinone combinatorial libraries and related products and methods for the treatment of disease SUGEN, INC. 2005-09-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050197382-A1 Indolinone combinatorial libraries and related products and methods for the treatment of disease FRK, PTK2, DSTYK LRRK2 289/4885PSEN1 3695/4885PSEN2 3641/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.