SCHEMBL5369931

SCHEMBL5369931

Cc1[nH]c(C)c(C(=O)O)c1Br

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.40
NOTUM Q6P988 2/20 0.40
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
NPSR1 Q6W5P4 2/20 0.35
TSHR P16473 1/20 0.35
LMNA P02545 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.33
MAPT P10636 1/20 0.33
PKM P14618 1/20 0.33
HSD17B10 Q99714 2/20 0.32
KDM4E B2RXH2 1/20 0.32
GAA P10253 1/20 0.32
HPGD P15428 1/20 0.32
GPR35 Q9HC97 2/20 0.32
ATM Q13315 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
POLB P06746 1/20 0.31
KMT2A Q03164 1/20 0.31
HCAR2 Q8TDS4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23147143 0.85 ALDH1A1 (0.37) ALDH1A1NOTUMCYP1A2CYP3A4NPSR1
SCHEMBL71362 0.82 NOTUM (0.48) ALDH1A1NOTUMCYP1A2CYP3A4NPSR1
SCHEMBL6468905 0.76 NPSR1 (0.52) ALDH1A1CYP1A2CYP3A4NPSR1TSHR
SCHEMBL11584471 0.75 ALDH1A1 (0.52) ALDH1A1NOTUMCYP1A2CYP3A4NPSR1
SCHEMBL11802081 0.75 NOTUM (0.43) ALDH1A1NOTUMCYP1A2CYP3A4NPSR1
SCHEMBL11223557 0.74 NOTUM (0.41) ALDH1A1NOTUMCYP1A2CYP3A4SMN1; SMN2
SCHEMBL7424028 0.73 CYP1A2 (0.52) ALDH1A1NOTUMCYP1A2CYP3A4NPSR1
SCHEMBL13154639 0.70 NOTUM (0.38) ALDH1A1NOTUMCYP1A2CYP3A4SMN1; SMN2
SCHEMBL5035539 0.70 GPR35 (0.46) ALDH1A1CYP1A2CYP3A4NPSR1TSHR
SCHEMBL29950777 0.70 SMN1; SMN2 (0.58) ALDH1A1NOTUMCYP1A2CYP3A4NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007145349-A2 SUBSTITUTED PYRROLE DERIVATIVES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-12-21 WO disclosed
EP-1466902-A1 ANDROGEN RECEPTOR ANTAGONISTS Takeda Chemical Industries, Ltd. (JP) 2004-10-13 EP disclosed
WO-1999001423-A1 GLUCAGON ANTAGONISTS/INVERSE AGONISTS NOVO NORDISK A/S (DK) 1999-01-14 WO disclosed