SCHEMBL5370041

SCHEMBL5370041

CON(C)C(=O)c1cn(-c2ccc(Cl)cc2)c(-c2ccc(Cl)cc2Cl)n1

nearest known ligand 0.56

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 17/20 0.56
CNR2 P34972 5/20 0.56
GABRA2 P47869 3/20 0.47
GABRB2 P47870 3/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6342475 0.89 CNR1 (0.67) CNR1CNR2GABRA2GABRB2
SCHEMBL674935 0.83 GABRA2 (0.67) CNR1CNR2GABRA2GABRB2
SCHEMBL5367435 0.82 CNR1 (0.64) CNR1CNR2GABRA2GABRB2
SCHEMBL4501902 0.81 CNR1 (0.65) CNR1CNR2GABRA2GABRB2
SCHEMBL4434578 0.81 CNR1 (0.65) CNR1CNR2GABRA2GABRB2
SCHEMBL4510387 0.80 CNR1 (0.54) CNR1CNR2GABRA2GABRB2
SCHEMBL4479830 0.80 GABRA2 (0.72) CNR1CNR2GABRA2GABRB2
SCHEMBL4474828 0.79 CNR1 (0.63) CNR1CNR2GABRA2GABRB2
SCHEMBL6332950 0.79 CNR1 (0.68) CNR1CNR2GABRA2GABRB2
SCHEMBL5370038 0.78 CNR1 (0.62) CNR1CNR2GABRA2GABRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070254935-A1 PYRAZOLE AND IMIDAZOLE COMPOUNDS AND USES THEREOF PFIZER, INC. 2007-11-01 US disclosed
US-7247628-B2 Cannabinoid receptor ligands and uses thereof PFIZER, INC. (US) 2007-07-24 US disclosed
EP-1572662-A1 PYRAZOLE AND IMIDAZOLE COMPOUNDS AND USES THEREOF Pfizer Products Inc. (US) 2005-09-14 EP disclosed
WO-2004052864-A1 PYRAZOLE AND IMIDAZOLE COMPOUNDS AND USES THEREOF PFIZER PRODUCTS INC. (US) 2004-06-24 WO disclosed
US-20040122074-A1 Cannabinoid receptor ligands and uses thereof PFIZER INC. 2004-06-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040122074-A1 Cannabinoid receptor ligands and uses thereof CNR1, CNR2, GPR18 CNR1 1/4885CNR2 2/4885GABRA2 41/4885
US-20070254935-A1 PYRAZOLE AND IMIDAZOLE COMPOUNDS AND USES THEREOF CNR2, CNR1, GPR18 CNR1 2/4885CNR2 1/4885GABRA2 26/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.