SCHEMBL5370156

SCHEMBL5370156

Nc1ncc(C(=O)NCC2CCN(S(=O)(=O)CCc3ccccc3)CC2)cn1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 7/20 0.51
FAAH O00519 1/20 0.48
HDAC3 O15379 6/20 0.45
HDAC4 P56524 6/20 0.45
HDAC1 Q13547 6/20 0.45
HDAC7 Q8WUI4 6/20 0.45
HDAC2 Q92769 6/20 0.45
HDAC10 Q969S8 6/20 0.45
HDAC11 Q96DB2 6/20 0.45
HDAC8 Q9BY41 6/20 0.45
HDAC9 Q9UKV0 6/20 0.45
HDAC5 Q9UQL6 6/20 0.45
F10 P00742 1/20 0.44
CYP2C19 P33261 1/20 0.43
CKS1B P61024 1/20 0.43
SKP1 P63208 1/20 0.43
SKP2 Q13309 1/20 0.43
LMNA P02545 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.42
FKBP1A P62942 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14425189 0.90 MEN1 (0.48) HDAC6F10LMNA
SCHEMBL14425184 0.88 HDAC6 (0.52) HDAC6FAAHHDAC3HDAC4HDAC1
SCHEMBL5363063 0.87 HDAC6 (0.52) HDAC6FAAHHDAC3HDAC4HDAC1
SCHEMBL5368614 0.85 HDAC6 (0.55) HDAC6FAAHHDAC3HDAC4HDAC1
SCHEMBL14425186 0.84 HDAC6 (0.51) HDAC6FAAHHDAC3HDAC4HDAC1
SCHEMBL5362714 0.83 HDAC6 (0.59) HDAC6FAAHHDAC3HDAC4HDAC1
SCHEMBL14425182 0.83 FAAH (0.49) HDAC6FAAHF10CYP2C19LMNA
SCHEMBL5359104 0.82 KDM4E (0.48) HDAC6FAAHF10CYP2C19CKS1B
SCHEMBL14425181 0.81 FAAH (0.49) HDAC6FAAHCYP2C19LMNASMN1; SMN2
SCHEMBL14425178 0.79 FAAH (0.49) HDAC6FAAHHDAC3HDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed