SCHEMBL5372889

SCHEMBL5372889

CCc1c(C(N)=O)cc(C)cc1C(N)=O

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.39
NNMT P40261 1/20 0.38
CD38 P28907 1/20 0.38
MAPK8 P45983 1/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
POLB P06746 1/20 0.37
PARP1 P09874 4/20 0.36
CDC7 O00311 1/20 0.36
CNR1 P21554 1/20 0.35
CNR2 P34972 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
PARP10 Q53GL7 1/20 0.35
DHODH Q02127 1/20 0.35
SIRT3 Q9NTG7 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13504652 0.92 KDM4E (0.37) KDM4ENNMTCD38MAPK8L3MBTL1
SCHEMBL1003868 0.90 KDM4E (0.44) KDM4ENNMTCD38MAPK8L3MBTL1
SCHEMBL27516124 0.80 KDM4E (0.50) KDM4ETDP1
SCHEMBL3351899 0.79 KDM4E (0.37) KDM4ENNMTCD38MAPK8L3MBTL1
SCHEMBL14604836 0.78 KDM4E (0.44) KDM4ENNMTMAPK8L3MBTL1POLB
SCHEMBL4951717 0.78 SMN1; SMN2 (0.39) KDM4ENNMTL3MBTL1POLBPARP1
SCHEMBL1521942 0.76 POLB (0.37) KDM4ENNMTL3MBTL1POLBPARP1
SCHEMBL6173916 0.76 PARP1 (0.43) CD38MAPK8PARP1
SCHEMBL45719 0.76 PARP1 (0.51) KDM4EPARP1CYP3A4
SCHEMBL6001788 0.75 ALDH1A1 (0.38) KDM4EPARP1CDC7SMN1; SMN2TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1453789-A2 N,N'-SUBSTITUTED-1,3-DIAMINO-2-HYDROXYPROPANE DERIVATIVES Elan Pharmaceuticals, Inc. (US) 2004-09-08 EP claimed
WO-2003040096-A2 N, N'-SUBSTITUTED-1,3-DIAMINO-2-HYDROXYPROPANE DERIVATIVES ELAN PHARMACEUTICALS, INC. (US) 2003-05-15 WO claimed
US-7176242-B2 N,N′-substituted-1,3-diamino-2-hydroxypropane derivatives ELAN PHARMACEUTICALS, INC. (US) 2007-02-13 US disclosed