SCHEMBL5373702

SCHEMBL5373702

Cc1c(Cc2ccc(Cl)c(Oc3cccc(Br)c3)c2)n[nH]c(=O)c1C

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 15/20 0.45
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
TSHR P16473 1/20 0.40
CYP2C19 P33261 1/20 0.40
PRMT5 O14744 2/20 0.39
WDR77 Q9BQA1 2/20 0.39
ADORA2A P29274 2/20 0.36
ADORA1 P30542 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5364878 0.86 PARP1 (0.43) PARP1CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL5377272 0.85 PRMT5 (0.43) PARP1CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL5374033 0.84 CYP3A4 (0.41) PARP1CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL4661620 0.83 PARP1 (0.38) PARP1CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL5374044 0.82 PARP1 (0.41) PARP1CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL5375576 0.79 PARP1 (0.39) PARP1CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL5373478 0.79 CYP3A4 (0.38) PARP1CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL5381953 0.79 CYP3A4 (0.38) PARP1CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL4807235 0.78 APOBEC3G (0.40) PARP1CYP3A4ADORA2AADORA1
SCHEMBL4810024 0.78 SLC22A12 (0.45) PARP1CYP3A4ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed