SCHEMBL5374044

SCHEMBL5374044

CN(C)c1cc(=O)[nH]nc1Cc1ccc(Cl)c(Oc2cccc(Br)c2)c1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 12/20 0.41
CYP3A4 P08684 2/20 0.38
CYP2C9 P11712 1/20 0.35
TSHR P16473 1/20 0.35
CYP2C19 P33261 1/20 0.35
HTR2A P28223 1/20 0.34
SLC6A4 P31645 1/20 0.34
KCNH2 Q12809 1/20 0.34
ADORA2A P29274 2/20 0.33
ADORA1 P30542 2/20 0.33
CCR5 P51681 1/20 0.33
FNTA P49354 1/20 0.32
FNTB P49356 1/20 0.32
PGGT1B P53609 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5364878 0.88 PARP1 (0.43) PARP1CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL5375576 0.85 PARP1 (0.39) PARP1CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL5364926 0.83 CYP3A4 (0.54) PARP1CYP3A4HTR2ASLC6A4KCNH2
SCHEMBL5373702 0.82 PARP1 (0.45) PARP1CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL5374033 0.78 CYP3A4 (0.41) PARP1CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL4807235 0.77 APOBEC3G (0.40) PARP1CYP3A4HTR2ASLC6A4KCNH2
SCHEMBL4810024 0.76 SLC22A12 (0.45) PARP1CYP3A4HTR2ASLC6A4KCNH2
SCHEMBL5373600 0.76 CYP3A4 (0.45) PARP1CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL5373462 0.76 CYP3A4 (0.41) PARP1CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL4800114 0.76 ICAM1 (0.36) PARP1CYP3A4HTR2ASLC6A4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed