SCHEMBL5375576

SCHEMBL5375576

CN(C)c1cc(Cc2ccc(Cl)c(Oc3cccc(Br)c3)c2)n[nH]c1=O

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 7/20 0.39
CYP3A4 P08684 2/20 0.37
HTR2A P28223 2/20 0.33
SLC6A4 P31645 2/20 0.33
KCNH2 Q12809 2/20 0.33
ADORA2A P29274 2/20 0.32
ADORA1 P30542 2/20 0.32
CYP2C9 P11712 1/20 0.32
TSHR P16473 1/20 0.32
CYP2C19 P33261 1/20 0.32
GRM4 Q14833 1/20 0.32
CCR5 P51681 1/20 0.32
FNTA P49354 1/20 0.32
FNTB P49356 1/20 0.32
PGGT1B P53609 1/20 0.32
DAO P14920 2/20 0.32
DHFR P00374 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5374033 0.87 CYP3A4 (0.41) PARP1CYP3A4HTR2ASLC6A4KCNH2
SCHEMBL5377396 0.86 CYP3A4 (0.41) CYP3A4HTR2ASLC6A4KCNH2CYP2C9
SCHEMBL5374044 0.85 PARP1 (0.41) PARP1CYP3A4HTR2ASLC6A4KCNH2
SCHEMBL5373478 0.84 CYP3A4 (0.38) PARP1CYP3A4HTR2ASLC6A4KCNH2
SCHEMBL5381953 0.84 CYP3A4 (0.38) PARP1CYP3A4HTR2ASLC6A4KCNH2
SCHEMBL5364926 0.82 CYP3A4 (0.54) PARP1CYP3A4HTR2ASLC6A4KCNH2
SCHEMBL14559703 0.81 CYP3A4 (0.42) PARP1CYP3A4HTR2ASLC6A4KCNH2
SCHEMBL14559738 0.80 THRA (0.31) PARP1CYP3A4CYP2C9CYP2C19DAO
SCHEMBL5368522 0.80 CYP3A4 (0.43) PARP1CYP3A4HTR2ASLC6A4KCNH2
SCHEMBL5373702 0.79 PARP1 (0.45) PARP1CYP3A4ADORA2AADORA1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed