SCHEMBL5373933

SCHEMBL5373933

Cc1ccc(Cc2ccc(=O)[nH]n2)cc1Cc1ccccc1Cl

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.45
AKR1B1 P15121 4/20 0.43
AR P10275 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.38
ADORA2A P29274 1/20 0.37
ADORA1 P30542 1/20 0.37
PDE3B Q13370 1/20 0.37
PDE3A Q14432 1/20 0.37
CYP2C19 P33261 1/20 0.36
HSD17B10 Q99714 1/20 0.36
DAO P14920 1/20 0.36
KDM4E B2RXH2 2/20 0.36
LMNA P02545 2/20 0.36
MAPT P10636 1/20 0.36
CNR2 P34972 1/20 0.35
ALDH1A1 P00352 1/20 0.35
PARP1 P09874 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5381870 0.85 CYP3A4 (0.48) CYP3A4AKR1B1ARDAOCNR2
SCHEMBL5374280 0.84 CYP3A4 (0.50) CYP3A4AKR1B1PDE3BPDE3AHSD17B10
SCHEMBL5368836 0.83 CYP3A4 (0.64) CYP3A4AKR1B1PDE3BPDE3ADAO
SCHEMBL5373848 0.83 CYP3A4 (0.54) CYP3A4ARHSD17B10KDM4EPARP1
SCHEMBL5382621 0.80 CYP3A4 (0.54) CYP3A4AKR1B1DAOALDH1A1
SCHEMBL5367073 0.79 CYP3A4 (0.44) CYP3A4AKR1B1ADORA2ACYP2C19KDM4E
SCHEMBL5386101 0.74 NR4A2 (0.47) CYP3A4AKR1B1
SCHEMBL5374344 0.74 CYP3A4 (0.43) CYP3A4AKR1B1CYP2C19
SCHEMBL5374337 0.73 CYP3A4 (0.47) CYP3A4AKR1B1CYP2C19
SCHEMBL5371246 0.72 CYP3A4 (0.48) CYP3A4ALDH1A1PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed