SCHEMBL5381870

SCHEMBL5381870

Cc1ccc(Cc2ccc(=O)[nH]n2)cc1Cc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.48
CNR2 P34972 1/20 0.41
GPR55 Q9Y2T6 1/20 0.41
POLB P06746 1/20 0.39
AKR1B1 P15121 1/20 0.39
DAO P14920 1/20 0.38
AR P10275 1/20 0.37
PARP1 P09874 1/20 0.36
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
CYP1A2 P05177 1/20 0.36
NOTUM Q6P988 1/20 0.35
LDHA P00338 1/20 0.35
LDHB P07195 1/20 0.35
LNPEP Q9UIQ6 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5374280 0.88 CYP3A4 (0.50) CYP3A4CNR2AKR1B1LDHALDHB
SCHEMBL5368836 0.88 CYP3A4 (0.64) CYP3A4AKR1B1DAO
SCHEMBL5373933 0.85 CYP3A4 (0.45) CYP3A4CNR2AKR1B1DAOAR
SCHEMBL5373848 0.85 CYP3A4 (0.54) CYP3A4ARPARP1NOTUM
SCHEMBL5382621 0.84 CYP3A4 (0.54) CYP3A4POLBAKR1B1DAOCYP1A2
SCHEMBL5351260 0.83 AKR1B1 (0.51) CYP3A4POLBAKR1B1DAOAR
SCHEMBL5371246 0.79 CYP3A4 (0.48) CYP3A4PARP1
SCHEMBL5370985 0.79 CYP3A4 (0.48) CYP3A4DAOPARP1
SCHEMBL18127144 0.77 PTGS1 (0.51) CYP3A4POLBDAOCYP1A2
SCHEMBL146770 0.76 CALM1 (0.50) CYP3A4LDHALDHB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed