SCHEMBL5374946

SCHEMBL5374946

O=c1ccc(Cc2ccc(C(F)(F)F)c(Oc3ccccc3Cl)c2)n[nH]1

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.42
AR P10275 1/20 0.38
KDR P35968 2/20 0.36
AKR1B1 P15121 2/20 0.35
NTRK1 P04629 1/20 0.35
SCN8A Q9UQD0 1/20 0.35
SCN10A Q9Y5Y9 1/20 0.35
KMT2A Q03164 1/20 0.34
DAO P14920 1/20 0.33
CAMK2A Q9UQM7 1/20 0.33
PRMT5 O14744 1/20 0.32
WDR77 Q9BQA1 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5374337 0.88 CYP3A4 (0.47) CYP3A4AKR1B1CAMK2APRMT5WDR77
SCHEMBL5377719 0.86 CYP3A4 (0.46) CYP3A4AKR1B1CAMK2APRMT5WDR77
SCHEMBL5366909 0.86 CYP3A4 (0.46) CYP3A4KDRAKR1B1NTRK1SCN8A
SCHEMBL5368699 0.85 AR (0.39) CYP3A4ARAKR1B1PRMT5WDR77
SCHEMBL5375034 0.84 CYP3A4 (0.37) CYP3A4ARKDRNTRK1DAO
SCHEMBL5377568 0.84 CYP3A4 (0.47) CYP3A4ARKDRSCN8ASCN10A
SCHEMBL5367073 0.84 CYP3A4 (0.44) CYP3A4AKR1B1CAMK2APRMT5WDR77
SCHEMBL5374482 0.83 CYP3A4 (0.61) CYP3A4ARKDRAKR1B1PRMT5
SCHEMBL5374344 0.83 CYP3A4 (0.43) CYP3A4AKR1B1CAMK2APRMT5WDR77
SCHEMBL5373947 0.79 CYP3A4 (0.44) CYP3A4AKR1B1DAOPRMT5WDR77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
EP-1608629-A1 BENZYL-PYRIDAZINONS AS REVERSE TRANSCRIPTASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-28 EP disclosed
US-20040198736-A1 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC 2004-10-07 US disclosed
WO-2004085406-A1 BENZYL-PYRIDAZINONS AS REVERSE TRANSCRIPTASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2004-10-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040198736-A1 Non-nucleoside reverse transcriptase inhibitors POLR1A, POLR2A, POLR2E CYP3A4 264/4885AR 2411/4885KDR 3798/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.