SCHEMBL5374515

SCHEMBL5374515

CCc1ccc2nc(C(=O)O)n(COCC[Si](C)(C)C)c(=O)c2c1C

nearest known ligand 0.38

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.37
KLKB1 P03952 1/20 0.35
F11 P03951 1/20 0.33
F2RL1 P55085 1/20 0.31
MAPT P10636 1/20 0.31
ELANE P08246 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5381357 0.87 NPC1 (0.35) NPC1KLKB1F2RL1
SCHEMBL5369563 0.80 ELANE (0.42) NPC1KLKB1F11MAPTELANE
SCHEMBL4935109 0.74 CASR (0.39) NPC1ELANE
SCHEMBL4935725 0.73 MMP13 (0.40) NPC1MAPT
SCHEMBL4932747 0.73 ELANE (0.43) NPC1ELANE
SCHEMBL4934889 0.70 SMN1; SMN2 (0.38) NPC1MAPT
SCHEMBL30889616 0.70 NPC1 (0.36) NPC1KLKB1F11MAPT
SCHEMBL3059529 0.70 NPC1 (0.40) NPC1KLKB1F11MAPT
SCHEMBL1314051 0.69 NPC1 (0.35) NPC1KLKB1F11MAPT
SCHEMBL1316068 0.69 NPC1 (0.35) NPC1KLKB1F11MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1740551-A1 HETEROCYCLIC AMIDE COMPOUND AND USE THEREOF AS AN MMP-13 INHIBITOR Takeda Pharmaceutical Company Limited (JP) 2007-01-10 EP disclosed
WO-2005105760-A1 HETEROCYCLIC AMIDE COMPOUND AND USE THEREOF AS AN MMP-13 INHIBITOR TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2005-11-10 WO disclosed